首页> 外国专利> 2-phenyl-3-azoilbenzotiofenos to increase thrombomodulin expression.

2-phenyl-3-azoilbenzotiofenos to increase thrombomodulin expression.

机译:2-苯基-3-azoilbenzotiofenos增加血栓调节蛋白表达。

摘要

A METHOD FOR INCREASING THROMBOMODULIN EXPRESSION UNDERSTANDING TO ADMINISTER A HUMAN IN THE NEED OF TREATMENT AN EFFECTIVE AMOUNT OF A COMPONENT THAT HAS FORMULA (I) WHERE R1 AND R3 ARE INDEPENDENTLY HYDROGEN-C3-C6) -CO OR CO-AR, WHERE AR IS OPTIONALLY REPLACED PHENYL; R2 IS SELECTED FROM THE GROUP CONSISTING OF PIRROLIDINE, HEXAMETILENEIMINE, AND PIPERIDINE; OR A PHARMACEUTICALLY ACCEPTABLE SALT OF YOUR SOLVENT. THE INVENTION ALSO INCLUDES A METHOD FOR INHIBITING A THROMBOTIC DISEASE OR EVENT THAT INCLUDES MANAGING A HUMAN IN THE NEED OF IT AN EFFECTIVE AMOUNT OF A FORMULA COMPONENT 1. THE INVENTION ALSO INCLUDES A METHOD FOR INCREASING PROPORTION C THAT INCLUDES THE ADMINISTRATION OF A COMPONENT OF FORMULA 1.
机译:一种根据需要治疗人类需要的有效量的增加组成部分的凝血酶的蛋白表达的方法(I)R1和R3独立于氢-C3-C6 -CO或CO-AR在哪里可选取代的苯; R 2选自吡咯烷,己二烯亚胺和哌啶;或您的溶剂的药用盐。本发明还包括一种用于抑制血栓性疾病或事件的方法,该方法或方法需要对人类有效量的配方组分1进行管理。本发明还包括一种用于增加比例C的方法,该方法包括对组分的管理。公式1。

著录项

  • 公开/公告号ES2180564T3

    专利类型

  • 公开/公告日2003-02-16

    原文格式PDF

  • 申请/专利权人 ELI LILLY AND COMPANY;

    申请/专利号ES19940309485T

  • 发明设计人 CALNEK DAVID SCOTT;GRINNELL BRIAN WILLIAM;

    申请日1994-12-19

  • 分类号A61K31/445;A61K31/40;A61K31/38;A61P7/02;

  • 国家 ES

  • 入库时间 2022-08-21 23:59:14

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