首页> 外国专利> DERIVATIVES OF FURANO- AND THIOPHEN-CARBOTIOAMIDE, ITS PREPARATION AND ITS USE AS INHIBITORS OF THE REPLICATION OF HIV-1 AND MUTANTS OF HIV-1.

DERIVATIVES OF FURANO- AND THIOPHEN-CARBOTIOAMIDE, ITS PREPARATION AND ITS USE AS INHIBITORS OF THE REPLICATION OF HIV-1 AND MUTANTS OF HIV-1.

机译:呋喃和噻吩-碳酰胺的衍生物,其制备及其作为抑制HIV-1和HIV-1突变的抑制剂。

摘要

FORMULA COMPOUNDS (I), WHERE X IS OO S. THE COMPOUNDS OF THIS INVENTION ARE USEFUL FOR THE INHIBITION OF THE REPLICATION OF THE MUTANTS AND THE INVERSE TRANSCRIPT (RT) OF THE VIRUS OF THE HUMAN IMMUNODEFICIENCY (HIV-1), IN VITRO AND IN VIVO. THE COMPOUNDS ARE USEFUL IN THE THERAPEUTIC OR PREVENTIVE TREATMENT OF DISEASES CAUSED BY MUTANTS OF HIV-1 AND RT, SUCH AS A PURCHASED IMMUNODEFICIENCY SYNDROME (AIDS).
机译:式(I)中的X是OO。本发明的化合物可用于体外抑制人类免疫缺陷病毒(HIV-1)病毒的复制和逆转录(RT)的复制和体内。该化合物可用于治疗或预防性治疗由多种HIV-1和RT引起的疾病,如购买的免疫缺陷综合症(艾滋病)。

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