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PROSTAGLANDIN F2Alpha ANALOGS AND THEIR USE IN COMBINATION WITH ANTIMICROBIAL PROTEINS FOR THE TREATMENT OF GLAUCOMA AND INTRAOCULAR HYPERTENSION
PROSTAGLANDIN F2Alpha ANALOGS AND THEIR USE IN COMBINATION WITH ANTIMICROBIAL PROTEINS FOR THE TREATMENT OF GLAUCOMA AND INTRAOCULAR HYPERTENSION
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机译:前列腺素F2α类似物及其与抗微生物蛋白结合治疗青光眼和眼内高压的应用
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摘要
An ophthalmic formulation for the treatment of glaucoma and intraocular pressure with a prostaglandin compound of the F-series (PGF), and particularly a prodrug form of a PGFSUB2alpha/SUB analog, such as an ester, amide, or internal lactone, wherein preservative is an antimicrobial peptide, such as lactoferrin. In particularly preferred embodiments, the prostaglandin compound is a macrocyclic internal 1,15-lactone, such as the 16-aryloxy prostaglandin analogs, illustratively fluprostenol or cloprstenol.
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