首页> 外国专利> 4-(6-FLUORO-1,2-BENZISOXAZOLYL)-1-PIPERIDINYL-PROPOXY-CHROMEN-4-ONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF PSYCHOSIS, SCHIZOPHRENIA AND ANXIETY

4-(6-FLUORO-1,2-BENZISOXAZOLYL)-1-PIPERIDINYL-PROPOXY-CHROMEN-4-ONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF PSYCHOSIS, SCHIZOPHRENIA AND ANXIETY

机译:4-(6-氟-1,2-苯并异恶唑基)-1-哌啶基-铬--4-酮衍生物,其制备及其在治疗精神分裂症,精神分裂症和焦虑症中的用途

摘要

The present invention relatesto 4-(6-fluoro-1,2-benzisoxazolyl)-1-piperidinyl-propoxy-chromen-4-onederivatives having formula (I),wherein R is hydrogen or alkylhaving 1 to 4 carbon atoms optionallysubstituted by hydroxyl, as well astheir pharmaceutically acceptableaddition salts, which are useful in thetreatment of psychosis, schizophreniaand anxiety.
机译:本发明涉及到4-(6-氟-1,2-苯并恶唑基)-1-哌啶基-丙氧基-铬烯-4-酮具有式(I)的衍生物,其中R是氢或烷基碳原子数为1-4的化合物被羟基取代,以及其药学上可接受的加成盐,在精神病,精神分裂症的治疗和焦虑。

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