首页> 外国专利> PREPARATION OF 3AR-3AA,4A,6A(R*),6AA-6-3-AMINO-4-1-(3-CHLORO-2-THIENYL)METHYLPROPYLAMINO-2-PYRIDINYLAMINO-N-ETHYLTETRAHYDRO-2,2-DIMETHYL-4H-CYCLOPENTA-1,3-DIOXOLE-4-CARBOXAMIDE, PREPARATION OF INTERMEDIATES THERETO, AND SAID INTERMEDIATES

PREPARATION OF 3AR-3AA,4A,6A(R*),6AA-6-3-AMINO-4-1-(3-CHLORO-2-THIENYL)METHYLPROPYLAMINO-2-PYRIDINYLAMINO-N-ETHYLTETRAHYDRO-2,2-DIMETHYL-4H-CYCLOPENTA-1,3-DIOXOLE-4-CARBOXAMIDE, PREPARATION OF INTERMEDIATES THERETO, AND SAID INTERMEDIATES

机译:制备[3AR- [3AA,4A,6A(R *),6AA]]-6-[[3-AMINO-4-[[1-[(3-氯-2-噻吩基)甲基]丙基]酰胺基] -2-吡啶基[氨基] -N-乙基四氢-2,2-二甲基-4H-环戊TA-1,3-二恶唑-4-羧酰胺,中间体的制备和所述中间体

摘要

This invention is directed to methods for the preparation of [1S-[1a, 2b,3b,4a(S*)] ]-4-[7-[[1-(3-chloro-2-thienyl)methyl]propyl]amino]-3H- imidazo[4,5-b]pyridin-3-yl]-N-ethyl-2, 3-dihydroxycyclopentanecarboxamide, methods for the preparation of intermediates thereto, and to said intermediates themselves.
机译:本发明涉及制备[1S- [1a,2b,3b,4a(S *)]]-4- [7-[[1-(3-氯-2-噻吩基)甲基]丙基]的方法。氨基] -3H-咪唑并[4,5-b]吡啶-3-基] -N-乙基-2,3-二羟基环戊烷羧酰胺,其中间体的制备方法,以及所述中间体本身。

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