首页> 外国专利> BENZOTIAZOLE DERIVATIVES AS Adenosine Receptor Ligands

BENZOTIAZOLE DERIVATIVES AS Adenosine Receptor Ligands

机译:苯并噻唑衍生物作为腺苷受体配体

摘要

This invention relates to compounds of formula I wherein RSUP1 /SUPand RSUP2 /SUPare defined herein, or a pharmaceutically acceptable salt thereof. It has been found that the compounds of formula I are adenosine receptor ligands with good affinity to the ASUB2A/SUB-receptor and a high selectivity to the ASUB1/SUB- and ASUB3 /SUBreceptors. These compounds are useful, inter alia, in treatment of Alzheimer's disease, depression, Parkinson's disease and ADHD.
机译:本发明涉及式I化合物或其药学上可接受的盐,其中本文定义了R 1 和R 2 。已经发现式I化合物是对A 2A -受体具有良好亲和力并且对A 1 -和A 3 个受体。这些化合物尤其可用于治疗阿尔茨海默氏病,抑郁症,帕金森氏病和ADHD。

著录项

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号