首页> 外国专利> TGF- SIGNAL TRANSMISSION MECHANISM INHIBITOR, SMAD DEGRADATION INDUCTOR, SMAD UBIQUITIN FORMATION PROMOTER, SMURF DEGRADATION INDUCTOR, SMURF UBIQUITIN FORMATION PROMOTER, METHOD FOR INHIBITING TGF- SIGNAL TRANSMISSION MECHANISM, METHOD FOR INDUCING SMAD DEGRADATION, METHOD FOR PROMOTING SMAD UBIQUITIN FORMATION, METHOD FOR INDUCING SMURF DEGRADATION, AND METHOD FOR PROMOTING SMURF UBIQUITIN FORMATION

TGF- SIGNAL TRANSMISSION MECHANISM INHIBITOR, SMAD DEGRADATION INDUCTOR, SMAD UBIQUITIN FORMATION PROMOTER, SMURF DEGRADATION INDUCTOR, SMURF UBIQUITIN FORMATION PROMOTER, METHOD FOR INHIBITING TGF- SIGNAL TRANSMISSION MECHANISM, METHOD FOR INDUCING SMAD DEGRADATION, METHOD FOR PROMOTING SMAD UBIQUITIN FORMATION, METHOD FOR INDUCING SMURF DEGRADATION, AND METHOD FOR PROMOTING SMURF UBIQUITIN FORMATION

机译:TGF-信号传导机制抑制剂,SMAD降解诱导剂,SMAB-泛素形成促进剂,SMURF降解诱导剂,SMURF-泛素形成促进剂,TGF-信号传导机理的抑制方法,诱导SMAD-SMAD的方法蔓延降解,以及促进蔓延泛素形成的方法

摘要

PROBLEM TO BE SOLVED: To provide a TGF- signal transmission mechanism inhibitor.;SOLUTION: An estrogen receptor ligand, a glucocorticoid receptor ligand, a vitamin D receptor ligand, a progesterone receptor ligand, or a retinoic acid receptor ligand is used as a TGF- signal transmission mechanism inhibitor. The TGF- signal transmission mechanism inhibitor is useful for treating and researching cancers (breast cancer, lung cancer, uterine cancer, prostatic cancer, pancreatic cancer, melanoma), pulmonary fibrosis, renal fibrosis, and hepatocirrhosis.;COPYRIGHT: (C)2008,JPO&INPIT
机译:解决的问题:提供一种TGF-信号传递机制抑制剂。解决方案:雌激素受体配体,糖皮质激素受体配体,维生素D受体配体,孕激素受体配体或视黄酸受体配体用作TGF -信号传输机制抑制剂。 TGF-信号传导机制抑制剂可用于治疗和研究癌症(乳腺癌,肺癌,子宫癌,前列腺癌,胰腺癌,黑色素瘤),肺纤维化,肾纤维化和肝硬化。; COPYRIGHT:(C)2008,日本特许厅

著录项

  • 公开/公告号JP2008174463A

    专利类型

  • 公开/公告日2008-07-31

    原文格式PDF

  • 申请/专利权人 ANKHS:KK;

    申请/专利号JP20070007436

  • 发明设计人 YANAGISAWA JUN;ICHIHARA NARIYASU;

    申请日2007-01-16

  • 分类号A61K45;A61K48;A61K38;A61K31/565;A61P1/16;A61P13/12;A61P11;A61P35;A61P35/04;A61P43;C12Q1/68;C12N5/10;G01N33/15;G01N33/50;C12N15/09;

  • 国家 JP

  • 入库时间 2022-08-21 20:23:19

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