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Enaminotiocarbonilicos substituted compounds for Combating animal parasites and processes for their Preparation

机译:用于对抗动物寄生虫的Enaminotiocarbonilicos取代的化合物及其制备方法

摘要

Substituted enaminothio compounds (I) are new, where (I) excludes 4-{[(6-chloropyrid-3-yl)methyl](methyl)amino}furan-2(5H)-thione, 4-{[(6-chloropyrid-3-yl)methyl]amino}furan-2(5H)-thione, 4-{[(6-chloropyrid-3-yl)methyl](methyl)amino}thiophen-2(5H)-thione and 4-{[(6-chloropyrid-3-yl)methyl](ethyl)amino}thiophen-2(5H)-thione. Substituted enaminothio compounds of formula (I) are new, where (I) excludes 4-{[(6-chloropyrid-3-yl)methyl](methyl)amino}furan-2(5H)-th ione, 4-{[(6-chloropyrid-3-yl)methyl]amino}furan-2(5H)-thione, 4-{[(6-chloropyrid-3-yl)methyl](methyl)amino}thiophen-2(5H)-thione and 4-{[(6-chloropyrid-3-yl)methyl](ethyl)amino}thiophen-2(5H)-thione. A : pyrid-2-yl, pyrid-4-yl or pyrid-3-yl (all optionally substituted in 6th-position by F, Cl, Br, CH 3, CF 3or CF 3O), pyridazin-3-yl (optionally substituted in 6-position by Cl or CH 3), or pyrazin-3-yl, 2-chloropyrazin-5-yl or 1,3-thiazol-5-yl (all optionally substituted in 2nd-position by Cl or CH 3), or pyrimidinyl, pyrazolyl, thiophenyl, oxazolyl, isoxazolyl, 1,2,4-oxadiazolyl, isothiazolyl, 1,2,4-triazolyl or 1,2,5-thiadiazolyl (all optionally substituted by F, Cl, Br, CN, NO 2, 1-4C-alkyl (optionally substituted by F and/or Cl), 1-3C-alkylthio (optionally substituted by F and/or Cl), or 1-3C-alkylsulfonyl (optionally substituted by F and/or Cl), or 1-3C-alkylsulfonyl (optionally substituted by F and/or Cl)), or pyridine group of formula (a); X : halo, alkyl or haloalkyl; Y 1halo, alkyl, haloalkyl, haloalkoxy, azido or CN; B 1O, S or methylene; R 1H, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, cycloalkyl, cyclodialkyl, halocycloalkyl, alkoxy or halocyclodialkyl; R 2H or halo; and R 3H or alkyl. [Image] [Image] - ACTIVITY : Pesticide; Arthropodicide; Insecticide; Arachnicide; Nematocide; Acaricide; Fungicide; Antibacterial; Virucide; Herbicide; Antimicrobial; Antifouling. - MECHANISM OF ACTION : None given.
机译:取代的烯氨基硫基化合物(I)是新的,其中(I)不包括4-{[((6-氯吡啶-3-基)甲基](甲基)氨基}呋喃-2(5H)-硫酮,4-{[((6-氯吡啶-3-基)甲基]氨基}呋喃-2(5H)-硫酮,4-{[((6-氯吡啶-3-基)甲基](甲基)氨基}噻吩-2(5H)-硫酮和4- {[((6-氯吡啶-3-基)甲基](乙基)氨基}噻吩-2(5H)-硫酮。式(I)的取代的烯氨基硫基化合物是新的,其中(I)不包括第4-{[((6-氯吡啶-3-基)甲基](甲基)氨基}呋喃-2(5H)-离子,4-{[ (6-氯吡啶-3-基)甲基]氨基}呋喃-2(5H)-硫酮,4-{[((6-氯吡啶-3-基)甲基](甲基)氨基}噻吩-2(5H)-硫酮和4-{[((6-氯吡啶-3-基)甲基](乙基)氨基}噻吩-2(5H)-硫酮。 A:吡啶-2-基,吡啶-4-基或吡啶-3-基(全部任选地在第6位被F,Cl,Br,CH 3,CF 3或CF 3O取代),哒嗪-3-基(任选地在6位上被Cl或CH 3取代)或吡嗪-3-基,2-氯吡嗪-5-基或1,3-噻唑-5-基(所有在2位上被Cl或CH 3取代)或嘧啶基,吡唑基,噻吩基,恶唑基,异恶唑基,1,2,4-恶二唑基,异噻唑基,1,2,4-三唑基或1,2,5-噻二唑基(均可选地被F,Cl,Br,CN, NO 2、1-4C-烷基(可选被F和/或Cl取代),1-3C-烷硫基(可选被F和/或Cl取代)或1-3C-烷基磺酰基(可选被F和/或Cl取代) )或1-3C-烷基磺酰基(任选地被F和/或Cl取代))或式(a)的吡啶基; X:卤素,烷基或卤代烷基; Y 1>卤代,烷基,卤代烷基,卤代烷氧基,叠氮基或CN; B 1> O,S或亚甲基; R 1> H,烷基,卤代烷基,烯基,卤代烯基,炔基,环烷基,环二烷基,卤代环烷基,烷氧基或卤代环二烷基; R 2> H或卤素; R 3> H或烷基。 [图像] [图像]-活动:农药;节肢动物杀菌剂;杀虫剂杀螨剂;杀线虫剂杀螨剂杀菌剂抗菌;杀病毒剂;除草剂;抗菌;防污。 -作用机理:未给出。

著录项

  • 公开/公告号CO6300829A2

    专利类型

  • 公开/公告日2011-07-21

    原文格式PDF

  • 申请/专利权人 BAYER CROPSCIENCE AG;

    申请/专利号CO20100117237

  • 申请日2010-09-22

  • 分类号A01N43/40;A01N43/78;C07D405/12;

  • 国家 CO

  • 入库时间 2022-08-21 18:06:55

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