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OLIGONUCLEOTIDES COUPLED WITH LIPID, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND THEIR USE IN INHIBITING TELOMERASE AND IN THE MANUFACTURE OF MEDICAMENTS FOR TREATING CANCER
OLIGONUCLEOTIDES COUPLED WITH LIPID, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND THEIR USE IN INHIBITING TELOMERASE AND IN THE MANUFACTURE OF MEDICAMENTS FOR TREATING CANCER
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机译:脂类与脂类,包含它们的药物组合物及其在抑制端粒酶和用于制备治疗癌症的药物中的用途
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摘要
Compounds comprising an oligonucleotide moiety covalently linked to a lipid moiety are disclosed. The oligonucleotide moiety comprises a sequence that is complementary to the RNA component of human telomerase. The compounds inhibit telomerase activity in cells with a high potency and have superior cellular uptake characteristics.
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