首页> 外国专利> (R) -3- (E) -2- (PYRR0LIDIN-3-YL) VINYL) -5- (TETRAHYDR0PYRAN-4-YL0XY) PYRIDINE, ITS SALTS, ITS SYNTHESIS AND ITS USE AS LIGAND FOR NICOTINIC ACETYLCHOLINERGIC RECEPTORS

(R) -3- (E) -2- (PYRR0LIDIN-3-YL) VINYL) -5- (TETRAHYDR0PYRAN-4-YL0XY) PYRIDINE, ITS SALTS, ITS SYNTHESIS AND ITS USE AS LIGAND FOR NICOTINIC ACETYLCHOLINERGIC RECEPTORS

机译:(R)-3-(E)-2-(PYRR0LIDIN-3-YL)乙烯基)-5-(TEHYDR0PYRAN-4-YL0XY)吡啶,其盐,其合成及其用作烟碱乙酰胆碱受体的配体

摘要

The present invention relates to the hemi-galactarate, oxalate and di-p-toluoyl-D-tartrate salt forms of (R)-3-((E)-2-(pyrrolidin-3-yl)vinyl)-5-(tetrahydropyran-4-yloxy)pyridine or hydrates or solvates thereof, compositions comprising these salt and their use for treating or preventing a NNR mediated disorder.
机译:本发明涉及(R)-3-((E)-2-(吡咯烷-3-基)乙烯基)-5-()的半半乳糖酸酯,草酸酯和二对甲苯甲酰基-D-酒石酸盐形式。四氢吡喃-4-基氧基)吡啶或其水合物或溶剂化物,包含这些盐的组合物及其在治疗或预防NNR介导的疾病中的用途。

著录项

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号