首页> 外国专利> ADMINISTRATION METHOD FOR PREPARATION CONTAINING OSELTAMIVIR CARBOXYLATE GUANIDINO ANALOGUES AND/OR ETHYL ESTERS THEREOF

ADMINISTRATION METHOD FOR PREPARATION CONTAINING OSELTAMIVIR CARBOXYLATE GUANIDINO ANALOGUES AND/OR ETHYL ESTERS THEREOF

机译:包含奥司他胺羧酸盐胍基类似物和/或乙基酯的制备方法

摘要

The present invention relates to an administration method for a preparation containing oseltamivir carboxylate guanidino analogues and/or ethyl esters thereof, the administration being carried out via inhalation. The present method treats colds caused by influenza viruses, and reduces dependence on a single type of drug, such as oseltamivir, zanamivir or peramivir, thereby preventing new resistant virus strains from being created due to widespread use of a single type. The present method also provides for the oseltamivir carboxylate guanidino analogues and/or ethyl esters thereof a method for greatly improving bioavailability compared with oral administration or intravenous drip injection. More importantly, the present method utilizes small doses, has fewer side effects and is fast-acting.
机译:本发明涉及含有奥司他韦羧酸盐胍基类似物和/或其乙酯的制剂的给药方法,该给药是通过吸入进行的。本方法治疗由流感病毒引起的感冒,并减少了对单一类型药物如奥司他韦,扎那米韦或帕拉米韦的依赖性,从而防止了由于单一类型的广泛使用而产生新的抗药性病毒株。本方法还为奥司他韦羧酸盐胍基类似物和/或其乙酯提供了一种与口服或静脉内滴注相比大大提高生物利用度的方法。更重要的是,本发明方法使用小剂量,副作用少并且作用迅速。

著录项

  • 公开/公告号WO2015027847A2

    专利类型

  • 公开/公告日2015-03-05

    原文格式PDF

  • 申请/专利权人 CHEN YONGQI;BAI ZHONGHU;DING YULONG;

    申请/专利号WO2014CN84835

  • 发明设计人 CHEN YONGQI;BAI ZHONGHU;DING YULONG;

    申请日2014-08-20

  • 分类号A61K31/215;A61K9/72;A61K9/12;A61K9/14;A61P31/16;A61P11;

  • 国家 WO

  • 入库时间 2022-08-21 15:08:02

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