首页> 外国专利> 5-ARYL OR 5-HETEROARYL SUBSTITUTED 3-HYDROXYPYRIDIN-2-YL-CARBONYLAMINO-ALKANOIC ACID DERIVATIVES AND SALTS THEREOF AS WELL AS THEIR PREPARATION FROM THE RESPECTIVE 3-HYDROXY-PICOLINIC ACID DERIVATIVES

5-ARYL OR 5-HETEROARYL SUBSTITUTED 3-HYDROXYPYRIDIN-2-YL-CARBONYLAMINO-ALKANOIC ACID DERIVATIVES AND SALTS THEREOF AS WELL AS THEIR PREPARATION FROM THE RESPECTIVE 3-HYDROXY-PICOLINIC ACID DERIVATIVES

机译:5-芳基或5-杂芳基取代的3-羟基吡啶-2-基-碳氨酯基-碱金属衍生物和其盐以及由相应的3-羟基-吡啶甲酸衍生物制备

摘要

The present invention relates to 5-aryl or 5-heteroaryl substituted 3-hydroxypyridin-2-yl-carbonylamino-alkanoic acid derivatives and salts thereof as well as to their preparation from the respective 3-hydroxy-picolinic acid derivatives. The final compounds are prolyl hydroxylase inhibitors.
机译:本发明涉及5-芳基或5-杂芳基取代的3-羟基吡啶-2-基-羰基氨基-链烷酸衍生物及其盐,以及由相应的3-羟基吡啶甲酸衍生物制备的方法。最终化合物是脯氨酰羟化酶抑制剂。

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