首页> 外国专利> APPLICATION OF SRC HOMOLOGY REGION 2-CONTAINING PROTEIN TYROSINE PHOSPHATASE-1 AGONIST FOR IMPROVING FIBROSIS

APPLICATION OF SRC HOMOLOGY REGION 2-CONTAINING PROTEIN TYROSINE PHOSPHATASE-1 AGONIST FOR IMPROVING FIBROSIS

机译:含蛋白酪氨酸磷酸酶-1蛋白的SRC同源区域2在改善纤维化中的应用

摘要

The present invention provides an application of an SRC homology region 2-containing tyrosine phosphatase-1 agonist in preparation of drugs for treating and reducing a fibrotic disease. Preferably, the agonist is formula (I) as represented by SC-43; the fibrotic disease is skin sclerosis, cardiac fibrosis, pulmonary fibrosis, hepatic fibrosis, pancreatic fibrosis, or renal fibrosis.
机译:本发明提供了含有SRC同源区2的酪氨酸磷酸酶-1激动剂在制备用于治疗和减轻纤维化疾病的药物中的应用。优选地,所述激动剂是由SC-43表示的式(I);纤维化疾病是皮肤硬化,心脏纤维化,肺纤维化,肝纤维化,胰腺纤维化或肾纤维化。

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