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Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

机译：在人组胺H4受体上评估组胺H1，H2-和H3受体配体：鉴定4-甲基组胺为第一个有效的选择性H4受体激动剂

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The histamine H

机译：组胺H

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Lim H.D.; van Rijn R.; Ling P.; Bakker R.A.; Thurmond R.L.; Leurs R.;
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年度 2005
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正文语种 eng
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1. Evaluation of Histamine H_1-,H_2-,and H_3-Receptor Ligands at the Human Histamine H_4 Receptor:Identification of 4-Methylhistamine as the First Potent and Selective H_4 Receptor Agonist [J] . Herman D.Lim, Richard M.van Rijn, Ping Ling, The Journal of Pharmacology and Experimental Therapeutics: Official Publication of the American Society for Pharmacology and Experimental Therapeutics . 2005,第3期

机译：人组胺H_4受体上组胺H_1-，H_2-和H_3-受体配体的评估：作为第一个有效和选择性H_4受体激动剂的4-甲基组胺的鉴定
2. Evaluation of Histamine H_1,-, H_2-, and H_3-Receptor Ligands at the Human Histamine H_4 Receptor: Identification of 4- Methylhistamine as the First Potent and Selective H_4 Receptor Agonist [J] . Herman D. Lim, Richard M. van Rijn, Ping Ling, The Journal of Pharmacology and Experimental Therapeutics: Official Publication of the American Society for Pharmacology and Experimental Therapeutics . 2005,第3期

机译：人组胺H_4受体上的组胺H_1，-，H_2-和H_3-受体配体的评估：4-甲基组胺作为第一个有效的选择性H_4受体激动剂的鉴定
3. Phenylalanine 169 in the second extracellular loop of the human histamine H4 receptor is responsible for the difference in agonist binding between human and mouse H4 receptors. [J] . Lim HD, Jongejan A, Bakker RA, The Journal of Pharmacology and Experimental Therapeutics: Official Publication of the American Society for Pharmacology and Experimental Therapeutics . 2008,第1期

机译：人组胺H4受体第二个胞外环中的苯丙氨酸169负责人和小鼠H4受体之间激动剂结合的差异。
4. Unraveling the Role of Histamine Receptors HI, H2, H3, and H4 in the Canine Gastrointestinal Tract [C] . Conference of the American College of Veterinary Internal Medicine (ACVIM) . 2017

机译：解开组胺受体HI，H 2，H3和H4在犬胃肠道中的作用
5. Novel mechanisms of cardioprotection: Catecholamine release by natriuretic peptides: Characterization and prevention; activation of ALDH2 in mast cell mitochondria: Prevention of local angiotensin II formation; activation of histamine H3-receptors: Reduction of angiotensin AT1-receptor neuronal expression [D] . Chan, Noel Yan-ki 2012

机译：心脏保护的新机制：利钠肽释放儿茶酚胺：表征和预防；肥大细胞线粒体中ALDH2的激活：预防局部血管紧张素II的形成； H3受体的活化：降低血管紧张素AT1受体神经元表达
6. Effects of histamine H1- H2- and H3-receptor selective drugs on the mechanical activity of guinea-pig small and large intestine. [O] . R. Leurs, M. M. Brozius, M. J. Smit, 1991

机译：组胺H1-H2-和H3-受体选择性药物对豚鼠小肠和大肠机械活性的影响。
7. N1-(3-Cyclohexylbutanoyl)-N2-3-(1H-imidazol-4-udyl)propylguanidine (UR-AK57), a Potent Partial Agonist for the Human Histamine H1- and H2- Receptors [O] . Xie Sheng-Xue, Kraus Anja, Ghorai Prasanta, 2006

机译：N1-（3-环己基丁酰基）-N2- 3-（1H-咪唑-4- ud）丙基胍（UR-AK57），一种有效的人类组胺H1-和H2-受体激动剂

Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

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