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Enantiospecific synthesis and pharmacological evaluation of a series of super-potent, conformationally restricted 5-HT(2A/2C) receptor agonists

机译：一系列超强效，构象限制的5-HT（2a / 2C）受体激动剂的对映特异性合成和药理学评价

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James J. Chambers; Deborah M. Kurrasch-orbaugh; Matthew A. Parker; David E. Nichols;
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年度 2015
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1. Enantiospecific synthesis and pharmacological evaluation of a series of super-potent, conformationally restricted 5-HT(2A/2C) receptor agonists. [J] . Chambers JJ, Kurrasch-Orbaugh DM, Parker MA, Journal of Medicinal Chemistry . 2001,第6期

机译：对映体的合成和一系列超强，构象受限的5-HT（2A / 2C）受体激动剂的药理学评价。
2. Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors. [J] . Knight AR, Misra A, Quirk K, Naunyn-Schmiedeberg's Archives of Pharmacology . 2004,第2期

机译：5-HT（2A），5-HT（2B）和5-HT（2C）受体激动剂放射性配体结合位点的药理学表征。
3. Conformationally constrained butyrophenones as new pharmacological tools to study 5-HT 2A and 5-HT 2C receptor behaviours. [J] . Brea J, Masaguer CF, Villazon M, European Journal of Medicinal Chemistry: Chimie Therapeutique . 2003,第4期

机译：构象受限的丁苯酮是研究5-HT 2A和5-HT 2C受体行为的新药理学工具。
4. Highly selective cyclic peptides for human melanocortin-4 receptor (MC-4):design,synthesis,bioactive conformation,and pharmacological evaluation as an anti-obesity agent [C] . Waleed Danho, Joseph Swistok, Adrian Cheung, the International Peptide Symposium . 2001

机译：用于人黑色素蛋白-4受体的高选择性环状肽（MC-4）：设计，合成，生物活性构象和作为抗肥胖剂的药理学评估
5. A 5-HT locomotor system: Identification, actions through 5-HT(2A/7) receptor subtypes, and effects on the control of locomotion. [D] . Liu, Jun. 2007

机译：5-HT运动系统：识别，通过5-HT（2A / 7）受体亚型的作用，以及对运动控制的影响。
6. A Novel Aminotetralin-Type Serotonin (5-HT) 2C Receptor-Specific Agonist and 5-HT2A Competitive Antagonist/5-HT2B Inverse Agonist with Preclinical Efficacy for Psychoses [O] . Clinton E. Canal, Drake Morgan, Daniel Felsing, -1

机译：具有精神病前临床疗效的新型氨基四氢萘型5-羟色胺（5-HT）2C受体特异性激动剂和5-HT2A竞争性拮抗剂/ 5-HT2B反向激动剂。
7. Design, Synthesis, and Evaluation of Proline and Pyrrolidine Based Melanocortin Receptor Agonists. A Conformationally Restricted Dipeptide Mimic Approach [O] . -1

机译：脯氨酸和吡咯烷基脲素受体激动剂的设计，合成和评价。一个综合限制的二肽模拟方法

Enantiospecific synthesis and pharmacological evaluation of a series of super-potent, conformationally restricted 5-HT(2A/2C) receptor agonists

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