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Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - neurokinin-1 antagonist peptidomimetics

机译：紧凑的，构象受限的双功能阿片类激动剂-Neurokinin-1拮抗剂拟肽的合成及生物学评价

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status: published

机译：状态：已发布

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Guillemyn Karel; Kleczkowska Patrycia; Lesniak Anna; Dyniewicz Jolanta; Van der Poorten Olivier; Van den Eynde Isabelle; Keresztes Attila; Varga Eva; Lai Josephine; Porreca Frank; Chung Nga; Lemieux Carole; Mika Joanna; Rojewska Ewelina; Makuch Wioletta; Van Duppen Joost; Przewlocka Barbara; Vanden Broeck Jozef; Lipkowski Andrzej; Schiller Peter; Tourwé Dirk; Ballet Steven;
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年度 2015
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1. Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - Neurokinin-1 antagonist peptidomimetics [J] . Guillemyn Karel, Kleczkowska Patrycia, Lesniak Anna, European Journal of Medicinal Chemistry: Chimie Therapeutique . 2015,第Null期

机译：紧凑的，构象受限的双功能阿片类激动剂-Neurokinin-1拮抗剂拟肽的合成和生物学评价
2. Design, synthesis, and biological evaluation of novel bifunctional C-terminal-modified peptides for delta/mu opioid receptor agonists and neurokinin-1 receptor antagonists [J] . Yamamoto T, Nair P, Davis P, Journal of Medicinal Chemistry . 2007,第12期

机译：设计，合成和生物学评估的新型双功能C末端修饰的肽为del / mu阿片受体激动剂和神经激肽1受体拮抗剂。
3. Synthesis and biological evaluation of new opioid agonist and neurokinin-1 antagonist bivalent ligands. [J] . Vardanyan R, Kumirov VK, Nichol GS, Bioorganic and medicinal chemistry . 2011,第20期

机译：新型阿片激动剂和神经激肽-1拮抗剂二价配体的合成和生物学评估。
4. Design, Synthesis and Biological Evaluation of Multivalent Ligands with μ/δ Opioid Agonist (μ-preferring) /NK-1 Antagonist Activities [C] . Aswini Kumar Giri, Qiong Xie, Christopher R. Apostol American Peptide Symposium . 2013

机译：多价配体的设计，合成和生物学评价，具有μ/δOpiOd激动剂（μ-opmoldring）/ NK-1拮抗剂活性
5. Synthesis and biological evaluation of conformationally constrained sphingosine-1-phosphate analogs as subtype selective S1P receptor agonist/antagonist. [D] . Zhu, Ran. 2008

机译：构象受限的鞘氨醇-1-磷酸类似物作为亚型选择性S1P受体激动剂/拮抗剂的合成和生物学评估。
6. Synthesis and biological evaluation of compact conformationally constrained bifunctional opioid agonist – neurokinin-1 antagonist peptidomimetics [O] . Karel Guillemyn, Patrycia Kleczkowska, Anna Lesniak, -1

机译：紧凑的构象受限的双功能阿片激动剂–神经激肽1拮抗剂拟肽的合成及生物学评价
7. The biological activity and metabolic stability of peptidic bifunctional compounds that are opioid receptor agonists and neurokinin-1 receptor antagonists with a cystine moiety [O] . Takashi Yamamoto, Padma Nair, Shou-wu Ma, 2009

机译：肽双官能化合物的生物活性和代谢稳定性，其是阿片受体激动剂和具有胱氨酸部分的神经喹啉-1受体拮抗剂

Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - neurokinin-1 antagonist peptidomimetics

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