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Structure-Activity Relationships within a Series of σ1 and σ2 Receptor Ligands: Identification of a σ2 Receptor Agonist (BS148) with Selective Toxicity against Metastatic Melanoma

机译：一系列Σ1和σ2受体配体中的结构 - 活性关系：鉴定σ2受体激动剂（BS148），具有抗转移性黑色素瘤的选择性毒性

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Silvia Franchini; Claudia Sorbi; Umberto Maria Battisti; Annalisa Tait; Leda Ivanova Bencheva; Elena Cichero; Paola Fossa; Antonio Cilia; Orazio Prezzavento; Simone Ronsisvalle; Giuseppina Aricò; Luisa Benassi; Cristina Vaschieri; Paola Azzoni; Cristina Magnoni; Livio Brasili;
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1. Structure-Activity Relationships within a Series of sigma(1) and sigma(2) Receptor Ligands: Identification of a sigma(2) Receptor Agonist (BS148) with Selective Toxicity against Metastatic Melanoma [J] . Franchini Silvia, Sorbi Claudia, Battisti Umberto Maria, ChemMedChem . 2017,第22期

机译：一系列Sigma（1）和Sigma（2）受体配体的结构 - 活性关系：鉴定σ（2）受体激动剂（BS148），具有针对转移性黑色素的选择性毒性
2. Structure-activity relationships of peptides incorporating a bioactive reverse-turn heterocycle at the melanocortin receptors: Identification of a 5800-fold mouse melanocortin-3 receptor (mMC3R) selective antagonist/partial agonist versus the mouse melanocortin-4 receptor (mMC4R) [J] . Singh A., Dirain M., Witek R., Journal of Medicinal Chemistry . 2013,第7期

机译：在黑皮质素受体上结合有生物活性反向杂环的肽的结构活性关系：鉴定5800倍小鼠黑皮质素-3受体（mMC3R）选择性拮抗剂/部分激动剂对小鼠黑皮质素4受体（mMC4R）
3. Structure-activity relationship-guided development of retinoic acid receptor-related orphan receptor gamma (RORγ)-selective inverse agonists with a phenanthridin-6(5H)-one skeleton from a liver X receptor ligand [J] . NishiyamaY., NakamuraM., MisawaT., Bioorganic and medicinal chemistry . 2014,第9期

机译：视黄酸受体相关的孤儿受体gamma（RORγ）选择性反向激动剂的结构-活性关系指导的发展，其具有来自肝脏X受体配体的phenanthridin-6（5H）-one骨架
4. Structure-activity relationship studies of new cyclic MSH analogues using cloned-human melanocortin receptors lead to greater selectivity and inverse agonists [C] . Minying Cai, Paolo Grieco, Jonathan Wiens, the International Peptide Symposium . 2001

机译：使用克隆人黑素激素受体的新循环MSH类似物的结构 - 活性关系研究导致更大的选择性和反向激动剂
5. Selective GLP-1 receptor antagonists and glucagon/GLP-1 co-agonists discovered through an investigation into the structure-activity relationship in glucagon-related peptides. [D] . Patterson, James T. 2011

机译：通过研究胰高血糖素相关肽的结构-活性关系，发现了选择性的GLP-1受体拮抗剂和胰高血糖素/ GLP-1共激动剂。
6. Structure-Activity Relationships of Peptides Incorporating a Bioactive Reverse-Turn Heterocycle at the Melanocortin Receptors: Identification of a 5800-fold Mouse Melanocortin-3 Receptor (mMC3R) Selective Antagonist/Partial Agonist versus the Mouse Melanocortin-4 Receptor (mMC4R) [O] . Anamika Singh, Marvin Dirain, Rachel Witek, -1

机译：在Melanocortin受体上掺入生物逆向杂环的肽的结构-活性关系：鉴定为5800倍小鼠Melanocortin-3受体（mMC3R）选择性拮抗剂/部分激动剂与小鼠Melanocortin-4受体（mMC4R）
7. Identification and Structure-Activity Relationship of Phenolic Acyl Hydrazones as Selective Agonists for the Estrogen-Related Orphan Nuclear Receptors ERRb and ERRg [O] . -1

机译：酚类酰基酰基腙作为雌激素相关孤儿核受体的选择性激动剂的鉴定和结构 - 活性关系errb和errg

Structure-Activity Relationships within a Series of σ1 and σ2 Receptor Ligands: Identification of a σ2 Receptor Agonist (BS148) with Selective Toxicity against Metastatic Melanoma

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