首页> 外文OA文献 >Two New Opioid Delta-Receptor Ligands: A Highly Selective Agon st and a Potent Selective Antagonist in in Vitro Isolated Preparations

【2h】

Two New Opioid Delta-Receptor Ligands: A Highly Selective Agon st and a Potent Selective Antagonist in in Vitro Isolated Preparations

机译：两种新的阿片类δ-受体配体：一种高度选择性的Agon St和体外分离制剂的强大有效的拮抗剂

代理获取

本网站仅为用户提供外文OA文献查询和代理获取服务，本网站没有原文。下单后我们将采用程序或人工为您竭诚获取高质量的原文，但由于OA文献来源多样且变更频繁，仍可能出现获取不到、文献不完整或与标题不符等情况，如果获取不到我们将提供退款服务。请知悉。

页面导航

著录项
引文网络
相似文献
相关主题

著录项

作者
Masaaki UEKI; Kazuko AOKI; Midori KAJIWARA; Kozo SHINOZAKI; Hideyuki INOUE; Tetsuo OKA;
展开▼
作者单位

展开▼
年度 1984
总页数
原文格式 PDF
正文语种
中图分类

相似文献

外文文献
中文文献
专利

1. Two New Opioid Delta-Receptor Ligands: A Highly Selective Agonist and a Potent Selective Antagonist in in Vitro Isolated Preparations [J] . Hideyuki INOUE, Kazuko AOKI, Kozo SHINOZAKI, Japanese Journal of Pharmacology . 1984,第4期

机译：两种新的阿片类药物δ受体配体：体外分离制剂中的高选择性激动剂和有效选择性拮抗剂。
2. DEVELOPMENT OF A MODEL FOR THE DELTA-OPIOID RECEPTOR PHARMACOPHORE .3. COMPARISON OF THE CYCLIC TETRAPEPTIDE, TYR-C[D-CYS-PHE-D-PEN]OH WITH OTHER CONFORMATIONALLY CONSTRAINED DELTA-RECEPTOR SELECTIVE LIGANDS [J] . Lomize AL., Mosberg HI., Pogozheva ID. Biopolymers: Original Research on Biomolecules and Biomolecular Assemblies . 1996,第2期

机译：三角洲阿片受体药物模型的开发3。环四肽TYR-C [D-CYS-PHE-D-PEN] OH与其他构象受约束的DELTA受体选择性配体的比较
3. Discovery of the First N-Substituted 4β-Methyl-5-(3-hydroxyphenyl)morphan To Possess Highly Potent and Selective Opioid δ Receptor Antagonist Activity [J] . F. Ivy Carroll, Li Zhang, S. WayneMascarella, Journal of Medicinal Chemistry . 2004,第2期

机译：发现第一个N-取代的4β-甲基-5-（3-羟苯基）吗啉具有高强度和选择性的阿片样物质δ受体拮抗剂活性。
4. Replacement of the Tyr~1 Hydroxyl Group of TIPP Peptides with N-(Alky)carboxamido Groups Results in Potent and Selective δ Opioid Agonists or Antagonists [C] . Irena Berezowska, Grazyna Weltrowska, Carole Lemieux American Peptide Symposium . 2009

机译：用N-（烷基）羧酰胺基团的TyR〜1羟基的Tyr〜1羟基导致有效和选择性的δ阿片类毒剂或拮抗剂
5. Synthesis towards salvinorin scaffold to develop a potential pain therapeutic and selective, potent kappa opioid ligands [D] . Strong, Tori Marquis 2012

机译：合成Salvinorin支架以开发潜在的止痛药和选择性，有效的阿片样物质配体
6. Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists. [O] . P W Schiller, T M Nguyen, G Weltrowska, 1992

机译：mu与delta类阿片受体对配体结合和信号转导的不同立体化学要求：一类有效且高度delta选择性的肽拮抗剂的开发。
7. Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists. [O] . Schiller, P W, Nguyen, T M, Weltrowska, G, 1992

机译：mu与delta类阿片受体对配体结合和信号转导的不同立体化学要求：一类有效且高度delta选择性的肽拮抗剂的开发。
8. Opioid Antagonist Properties of CTP, a Somatostatin Analog: In vivo Selectivity for Micron-Directed Ligands. [R] . Tortella, F. C., Echevarria, E., Holaday, J. W., 1989

机译：生长抑素类似物CTp的阿片拮抗剂性质：微定向配体的体内选择性。

Two New Opioid Delta-Receptor Ligands: A Highly Selective Agon st and a Potent Selective Antagonist in in Vitro Isolated Preparations

著录项

引文网络

相似文献

相关主题

期刊订阅