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Synthesis of Conformationally Restricted Analogs of Baclofen, a Potent GABAB Receptor Agonist, by the Introduction of a Cyclopropane Ring.

机译：通过引入环丙烷环来合成Baclofen，一种有效的荷兰受体激动剂的Baclofen的类似物。

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Satoshi SHUTO; Nobuko SHIBUYA; Shizuo YAMADA; Takashi OHKURA; Ryohei KIMURA; Akira MATSUDA;
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年度 1999
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1. Synthesis of conformationally restricted analogs of baclofen, a potent GABAB receptor agonist, by the introduction of a cyclopropane ring. [J] . Shuto S, Shibuya N, Yamada S, Chemical and Pharmaceutical Bulletin . 1999,第8期

机译：通过引入环丙烷环，合成强效GABA B受体激动剂巴氯芬构象受限的类似物。
2. Synthesis and structural and pharmacological properties of cyclopropane-based conformationally restricted analogs of 4-methylhistamine as histamine H3/H4 receptor ligands. [J] . Kobayashi T, Watanabe M, Yoshida Bioorganic and medicinal chemistry . 2010,第3期

机译：基于环丙烷的构象受限的4-甲基组胺作为组胺H3 / H4受体配体的合成及其结构和药理特性。
3. Design, Synthesis, and Evaluation of Conformationally Restricted Acetanilides as Potent and Selective β_3 Adrenergic Receptor Agonists for the Treatment of Overactive Bladder [J] . Christopher R. Moyes, Richard Berger, Stephen D. Goble, Journal of Medicinal Chemistry . 2014,第4期

机译：设计，合成和评价构象受限的乙酰苯胺作为有效和选择性β_3肾上腺素能受体激动剂治疗膀胱过度活动症
4. Synthesis and pharmacological activity of Dmt-Tic analogs with highly potent agonist and antagonist/agonist opioid activity [C] . Remo Guerrini, Gianfranco Balboni, Daniela Girolamo Calo, the International Peptide Symposium . 2001

机译：具有高效激动剂和拮抗剂/激动剂阿片类能活性DMT-TIC类似物的合成与药理活性
5. Synthesis and biological evaluation of conformationally constrained sphingosine-1-phosphate analogs as subtype selective S1P receptor agonist/antagonist. [D] . Zhu, Ran. 2008

机译：构象受限的鞘氨醇-1-磷酸类似物作为亚型选择性S1P受体激动剂/拮抗剂的合成和生物学评估。
6. Antitussive effects of the peripherally restricted GABAB receptor agonist lesogaberan in guinea pigs: comparison to baclofen and other GABAB receptor-selective agonists [O] . Brendan J Canning, Nanako Mori, Anders Lehmann 2012

机译：周围受限的GABA B受体激动剂来沙伯甘醇对豚鼠的镇咳作用：与巴氯芬和其他GABA B受体选择性激动剂的比较
7. Enantiospecific synthesis and pharmacological evaluation of a series of super-potent, conformationally restricted 5-HT(2A/2C) receptor agonists [O] . James J. Chambers, Deborah M. Kurrasch-orbaugh, Matthew A. Parker, 2015

机译：一系列超强效，构象限制的5-HT（2a / 2C）受体激动剂的对映特异性合成和药理学评价

Synthesis of Conformationally Restricted Analogs of Baclofen, a Potent GABAB Receptor Agonist, by the Introduction of a Cyclopropane Ring.

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