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Identification of Opioid Ligands Possessing Mixed μ Agonist/δ Antagonist Activity among Pyridomorphinans Derived from Naloxone, Oxymorphone, and Hydromorphone.

机译：鉴别纳洛酮，氧化甘油酮，氧化酮和氢酮酮吡啶卟啉烷烃中具有混合μ激动剂/δ拮抗剂活性的阿片类化合物的鉴定。

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Subramaniam Ananthan; Naveen K. Khare; Surendra K. Saini; Lainne E. Seitz; Jeffrey L. Bartlett; Peg Davis; Christina M. Dersch; Frank Porreca; Richard B. Rothman; Edward J. Bilsky;
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年度 2004
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1. Identification of Opioid Ligands Possessing Mixed μ Agonist/δ Antagonist Activity among Pyridomorphinans Derived from Naloxone, Oxymorphone, and Hydropmorphone [J] . Subramaniam Ananthan, Naveen K. Khare, Surendra K. Saini, Journal of Medicinal Chemistry . 2004,第6期

机译：纳洛酮，羟吗啡酮和氢吗啡酮衍生的吡吗啉中具有μ激动剂/δ混合拮抗剂活性的阿片类药物配体的鉴定
2. Discovery of tripeptide-derived multifunctional ligands possessing delta/mu opioid receptor agonist and neurokinin 1 receptor antagonist activities [J] . Nair Padma, Yamamoto Takashi, Cowell Scott, Bioorganic and Medicinal Chemistry Letters . 2015,第17期

机译：发现具有δ/μ阿片样物质受体激动剂和神经激肽1受体拮抗剂活性的三肽衍生的多功能配体
3. Synthesis and Structure-Activity Relationships of 5 '-Aryl-14-alkoxypyridomorphinans: Identification of a mu Opioid Receptor Agonist/delta Opioid Receptor Antagonist Ligand with Systemic Antinociceptive Activity and Diminished Opioid Side Effects [J] . Vekariya Rakesh H., Lei Wei, Ray Abhisek, Journal of Medicinal Chemistry . 2020,第14期

机译：5' - 14-烷氧基吡啶啉甲胺的合成及结构 - 活性关系：具有全身性抗血汗活性的MU阿片受体激动剂/三醇阿片受体受体拮抗剂配体的鉴定，并减少阿片类药物副作用
4. Identification of opioid receptor ligand interactions using structurally related delta-opioid receptor agonists and antagonists and molecular modeling. [C] . Sharon D.Bryant, Yunden Jinsmaa, Lawrence H.Lazarus International Peptide Symposium;European Peptide Symposium . 2005

机译：使用结构相关的δ-阿片类受体激动剂和拮抗剂和分子建模鉴定阿片受体配体的相互作用。
5. Ligand-based drug design: I. conformational studies of GBR 12909 analogs as cocaine antagonists; II. Three-dimensional-QSAR studies of salvinorin A analogs as kappa opioid agonists [D] . Pandit, Deepangi 2007

机译：基于配体的药物设计：I. GBR 12909类似物作为可卡因拮抗剂的构象研究；二。 Salvinorin A类似物作为κ阿片类激动剂的三维QSAR研究
6. Discovery of tripeptide-derived multifunctional ligands possessing delta/mu opioid receptor agonist and neurokinin 1 receptor antagonist activities [O] . Padma Nair, Takashi Yamamoto, Scott Cowell, -1

机译：发现具有δ/μ阿片样物质受体激动剂和神经激肽1受体拮抗剂活性的三肽衍生的多功能配体
7. Pyrrolo- and pyridomorphinans:Non-selective opioid antagonists and delta opioid agonists/mu opioid partial agonists [O] . Kumar, V., Clark, M.J., Traynor, J.R., 2014

机译：吡咯和吡ido吗啡：非选择性阿片拮抗剂和δ阿片激动剂/μ阿片部分激动剂
8. Opioid Antagonist Properties of CTP, a Somatostatin Analog: In vivo Selectivity for Micron-Directed Ligands. [R] . Tortella, F. C., Echevarria, E., Holaday, J. W., 1989

机译：生长抑素类似物CTp的阿片拮抗剂性质：微定向配体的体内选择性。

Identification of Opioid Ligands Possessing Mixed μ Agonist/δ Antagonist Activity among Pyridomorphinans Derived from Naloxone, Oxymorphone, and Hydromorphone.

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