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Muscarinic agonist, (±)-quinuclidin-3-yl-(4-fluorophenethyl)(phenyl)carbamate: High affinity, but low subtype selectivity for human M1 – M5 muscarinic acetylcholine receptors

机译：毒蕈碱激动剂，（±）-quinuclidin-3-Y1-（4-氟苯甲基）（苯基）氨基甲酸酯：高亲和力，但人体M1 - M5毒蕈碱乙酰胆碱受体的低亚型选择性

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Na-Ra Lee; Satheesh Gujarathi; Shobanbabu Bommagani; Kiranbabu Siripurapu; Guangrong Zheng; Linda P. Dwoskin;
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1. Muscarinic agonist, ( +/- )-quinuclidin-3-yl-(4-fluorophenethyl)(phenyl) carbamate: High affinity, but low subtype selectivity for human M-1 - M-5 muscarinic acetylcholine receptors [J] . Lee Na-Ra, Gujarathi Satheesh, Bommagani Shobanbabu, Bioorganic and Medicinal Chemistry Letters . 2019,第3期

机译：毒蕈碱激动剂，（+/-）-quinuclidin-3-基 - （4-氟苯乙基）（苯基）氨基甲酸酯：高亲和力，但人M-1-M-5毒蕈碱乙酰胆碱受体的低亚型选择性
2. Effects of imidafenacin (KRP-197/ONO-8025), a new anti-cholinergic agent, on muscarinic acetylcholine receptors. High affinities for M3 and M1 receptor subtypes and selectivity for urinary bladder over salivary gland. [J] . Kobayashi F, Yageta Y, Segawa M, Arzneimittel-Forschung: =Drug Research . 2007,第2期

机译：新型抗胆碱药伊达非那星（KRP-197 / ONO-8025）对毒蕈碱型乙酰胆碱受体的影响。 M3和M1受体亚型的高亲和力和唾液腺对膀胱的选择性。
3. Synthesis and SAR studies of 1,4-diazabicyclo(3.2.2)nonane phenyl carbamates--subtype selective, high affinity alpha7 nicotinic acetylcholine receptor agonists. [J] . ODonnell CJ, Peng L, ONeill BT Bioorganic and Medicinal Chemistry Letters . 2009,第16期

机译：1,4-二氮杂双环（3.2.2）壬烷苯基氨基甲酸酯的合成和SAR研究-亚型选择性高亲和力α7烟碱乙酰胆碱受体激动剂。
4. Cholinergic Modulation of CA1 Pyramidal Cells via M1 Muscarinic Receptor Activation: A Computational Study at Physiological and Supraphysiological Levels [C] . Adam R. Mergenthal, Jean-Marie C. Bouteiller, Theodore W. Berger Annual International Conference of the IEEE Engineering in Medicine and Biology Society . 2018

机译：通过M1毒蕈碱受体激活对CA1锥体细胞的胆碱能调节：生理和超生理水平的计算研究。
5. M1 muscarinic acetylcholine receptor regulation of endogenous transient receptor potential-canonical, subtype 6 (TRPC6) channels. [D] . Kim, Ju Young. 2005

机译：M1毒蕈碱型乙酰胆碱受体调节内源性瞬时受体电位-典型亚型6（TRPC6）通道。
6. Multiple Muscarinic Acetylcholine Receptor Subtypes Modulate Striatal Dopamine Release as Studied with M1–M5 Muscarinic Receptor Knock-Out Mice [O] . Weilie Zhang, Masahisa Yamada, Jesus Gomeza, 2002

机译：M1–M5毒蕈碱受体敲除小鼠研究多种毒蕈碱型乙酰胆碱受体亚型调节纹状体多巴胺释放
7. Involvement of a Subpopulation of Neuronal M4 Muscarinic Acetylcholine Receptors in the Antipsychotic-like Effects of the M1/M4 Preferring Muscarinic Receptor Agonist Xanomeline [O] . D. Dencker, G. Wortwein, P. Weikop, 2011

机译：在M1 / M4偏爱毒蕈碱受体激动剂Xanomeline的抗精神病的抗精神病的抗精神病患者中的脱硫症状的抗精神病患者血管蛋白受体中的介入
8. Short-Term Desensitization of Muscarinic Cholinergic Receptors in Mouse Neuroblastoma Cells: Selective Loss of Agonist Low-Affinity and Pirenzepine High-Affinity Binding Sites [R] . Cioffi, C. L., El-Fakahany, E. E. 1986

机译：小鼠神经母细胞瘤细胞中毒蕈碱胆碱能受体的短期脱敏：激动剂低亲和力和哌仑西平高亲和力结合位点的选择性丧失

Muscarinic agonist, (±)-quinuclidin-3-yl-(4-fluorophenethyl)(phenyl)carbamate: High affinity, but low subtype selectivity for human M1 – M5 muscarinic acetylcholine receptors

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