Investigations of new lead structures for the design of novel cyclooxygenase-2 inhibitors.

Park CH; Siomboing X; Yous S; Gressier B; Luyckx M; Chavatte P

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Investigations of new lead structures for the design of novel cyclooxygenase-2 inhibitors.

机译：用于设计新型环氧合酶2抑制剂的新型铅结构的研究。

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摘要

On the basis of molecular modelling studies, five new compounds were synthesised and studied in an attempt to design new lead structures as selective COX-2 inhibitors.

机译：在分子建模研究的基础上，合成并研究了五种新化合物，以尝试设计新的先导结构作为选择性COX-2抑制剂。

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来源
《European Journal of Medicinal Chemistry: Chimie Therapeutique》 |2002年第6期|共8页
作者
Park CH; Siomboing X; Yous S; Gressier B; Luyckx M; Chavatte P;
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原文格式 PDF
正文语种 eng
中图分类医药、卫生;
关键词
inhibitors; Lead; novel; Investigations; cyclooxygenase 2; 铅;

机译：抑制剂;铅;新颖;研究;环氧合酶2;铅;

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机译：用于设计新型环氧合酶2抑制剂的新型铅结构的研究。
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Investigations of new lead structures for the design of novel cyclooxygenase-2 inhibitors.

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