In vitro PAI-1 inhibitory activity of oxalamide derivatives.

Jain MR; Shetty S; Chakrabarti G; Pandya V; Sharma A; Parmar B; Srivastava S; Raviya M; Soni H; Patel PR

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In vitro PAI-1 inhibitory activity of oxalamide derivatives.

机译：草酰胺衍生物的体外PAI-1抑制活性。

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A number of oxalamide derivatives have been synthesized and evaluated for PAI-1 inhibitory activity. In vitro PAI-1 inhibitory activities of oxalamide derivatives are evaluated by chromogenic assay. Few compounds have shown significant PAI-1 inhibitory activity.

机译：已经合成了许多草酰胺衍生物，并评估了其对PAI-1的抑制活性。草酰胺衍生物的体外PAI-1抑制活性通过显色测定来评估。很少有化合物显示出显着的PAI-1抑制活性。

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《European Journal of Medicinal Chemistry: Chimie Therapeutique》 |2008年第4期|共5页
作者
Jain MR; Shetty S; Chakrabarti G; Pandya V; Sharma A; Parmar B; Srivastava S; Raviya M; Soni H; Patel PR;
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正文语种 eng
中图分类医药、卫生;劳动卫生;
关键词
Plasminogen Activator Inhibitor 1; derivatives; assay; Few; 纤溶酶原激活物抑制物1;

机译：Plasminogen Activator Inhibitor 1;derivatives;assay;Few;纤溶酶原激活物抑制物1;

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1. In vitro PAI-1 inhibitory activity of oxalamide derivatives. [J] . Jain MR, Shetty S, Chakrabarti G, European Journal of Medicinal Chemistry: Chimie Therapeutique . 2008,第4期

机译：草酰胺衍生物的体外PAI-1抑制活性。
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In vitro PAI-1 inhibitory activity of oxalamide derivatives.

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