机译:Human sirtuin 2 inhibitors, their mechanisms and binding modes
Universidade de Sao Paulo,Univ Sao Paulo;
Sch Pharmaceut Sci Ribeirao Preto,Univ Sao Paulo;
drug design; enzyme inhibition; enzyme inhibitory mechanisms; epigenetics; histone deacetylases; hSIRT2; HDAC; ligand binding modes; lysine deacetylases; sirtuin 2; STRUCTURAL BASIS; ADIPOCYTE DIFFERENTIATION; HISTONE DEACETYLASE; TERNARY COMPLEXES; CRYSTAL-STRUCTURE; ADP-RIBOSE; POTENT; SELECTIVITY; INSIGHTS; NAD(+);