...
机译:In Silico-Guided Rational Drug Design and Synthesis of Novel 4-(Thiophen-2-yl)butanamides as Potent and Selective TRPV1 Agonists
Univ Siena;
Magna Graecia Univ Catanzaro;
Univ CalabriaUniv Campania L VanvitelliCNRRecipharm Edmond Pharm;
STRUCTURE-AFFINITY RELATIONSHIPS; CAPSAICIN RECEPTOR TRPV1; VANILLOID TYPE-1 TRPV1; PHARMACOLOGICAL CHARACTERIZATION; ION-CHANNEL; LIGAND; RESINIFERATOXIN; BINDING; IDENTIFICATION; ACTIVATION;