机译:Potent macrocycle inhibitors of the human SAGA deubiquitinating module
Johns Hopkins Univ;
Univ Tokyo;
HISTONE H2B UBIQUITYLATION; TRANSCRIPTIONAL ACTIVATION; STRUCTURAL BASIS; NUCLEOSOME ACETYLATION; GENE-TRANSCRIPTION; TUMOR-SUPPRESSOR; DNA-REPAIR; COMPLEX; UBIQUITINATION; METHYLATION;