机译:基于片段的新型颠型Mek1粘合剂的发现
Structure Biophysics &
Fragments Discovery Sciences R&
D;
Structure Biophysics &
Fragments Discovery Sciences R&
D AstraZeneca;
Medicinal Chemistry Research &
Early Development Respiratory &
Immunology BioPharmaceuticals R&
D AstraZeneca;
Structure Biophysics &
Fragments Discovery Sciences R&
D;
Structure Biophysics &
Fragments Discovery Sciences R&
D AstraZeneca;
Discovery Biology Discovery Sciences R&
D AstraZeneca;
Structure Biophysics &
Fragments Discovery Sciences R&
D AstraZeneca;
Mechanistic Biology and Profiling Discovery Sciences R&
D AstraZeneca;
Medicinal Chemistry Research &
Early Development Respiratory &
Immunology BioPharmaceuticals R&
D AstraZeneca;
Medicinal Chemistry Research &
Early Development Respiratory &
Immunology BioPharmaceuticals R&
D AstraZeneca;
Structure Biophysics &
Fragments Discovery Sciences R&
D AstraZeneca;
Structure Biophysics &
Fragments Discovery Sciences R&
D AstraZeneca;
Medicinal Chemistry Research &
Early Development Respiratory &
Immunology BioPharmaceuticals R&
D AstraZeneca;
Structure Biophysics &
Fragments Discovery Sciences R&
D;
Structure Biophysics &
Fragments Discovery Sciences R&
D AstraZeneca;
MEK1; Kinases; Allosteric; COPD; Fragments; FBDD;
机译:MEK1的变构调节剂:药物设计和发现
机译:发现双功能致癌性靶向抑制剂的变构丝裂原激活的蛋白激酶(MEK1)和磷脂酰肌醇3-激酶(PI3K)。
机译:Caspase-7的变构调整:基于片段的药物发现方法
机译:用基于片段的药物设计和分子对接方法鉴定天然产物作为登革热病毒包膜蛋白β-OG口袋粘合剂的抑制剂
机译:ATCUN主题作为基于碎片的药物发现中的顺磁灯泡
机译:发现双功能致癌性靶向变应性丝裂原活化的蛋白激酶(MEK1)和磷脂酰肌醇3-激酶(PI3K)的抑制剂。
机译:用基于片段的药物设计和分子对接方法鉴定天然产物作为登革热病毒包膜蛋白β-OG口袋粘合剂的抑制剂
机译:导致体内肿瘤细胞死亡