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机译:双函数小分子抑制剂的靶向Bcl-2同源性3结构域并促进MCL-1泛素的失活
Dalian Univ Technol Zhang Dayu Sch Chem State Key Lab Fine Chem Dalian Liaoning Peoples R China;
Dalian Univ Technol Sch Chem Dalian Liaoning Peoples R China;
Dalian Univ Technol Sch Life Sci &
Technol Dalian Peoples R China;
Chinese Acad Sci Qingdao Inst Bioenergy &
Bioproc Technol Shandong Key Lab Synthet Biol Key Lab Biofuels Qingdao Shandong Peoples R China;
Dalian Univ Technol Sch Life Sci &
Technol Dalian Peoples R China;
Dalian Univ Technol Sch Chem Dalian Liaoning Peoples R China;
Chinese Acad Sci Inst Oceanol Qingdao Shandong Peoples R China;
Dalian Univ Technol Sch Chem Dalian Liaoning Peoples R China;
Dalian Univ Technol Sch Chem Dalian Liaoning Peoples R China;
apoptosis; conformation analysis; drug design; inhibitors; structure elucidation;
机译:双函数小分子抑制剂的靶向Bcl-2同源性3结构域并促进MCL-1泛素的失活
机译:通过靶向pleckstrin同源结构域并促进Akt泛素化的小分子抑制剂使Akt失活
机译:| [lsquo] |种子| [rsquo] |脱靶siRNA的分析揭示了Mcl-1在抵抗小分子Bcl-2 | [sol] | Bcl-XL抑制剂ABT-737中的重要作用
机译:一种新型的小分子IAP拮抗剂AZD5582,通过靶向CIAP1和XIAP在人胰腺癌中诱导诱导细胞凋亡的MCL-1下调
机译:热休克蛋白70通过防止抗凋亡的Bcl-2家族蛋白Mcl-1的蛋白酶体降解来抑制热诱导的细胞凋亡。
机译:通过靶向pleckstrin同源结构域并促进Akt泛素化的小分子抑制剂使Akt失活
机译:标准物:通过双函数小分子抑制剂去激活MCL-1,靶向BCL-2同源性3结构域并促进MCL-1泛素(Angew.Chem.46/2016)