首页> 外文期刊>Journal of Ethnopharmacology: An Interdisciplinary Journal Devoted to Bioscientific Research on Indigenous Drugs >Evaluation of the impact of Polygonum capitatum, a traditional Chinese herbal medicine, on rat hepatic cytochrome P450 enzymes by using a cocktail of probe drugs
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Evaluation of the impact of Polygonum capitatum, a traditional Chinese herbal medicine, on rat hepatic cytochrome P450 enzymes by using a cocktail of probe drugs

机译:用探针药物鸡尾酒评估一种传统的中草药,一种中草药,一种传统的中草药的影响较大的中草药肝细胞色素P450酶的影响

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摘要

Ethnopharmacological relevance: Polygonum capitatum is a well-known Miao medicinal plant that has been used for many years for its unique therapeutic effects on various urological disorders, including urinary calculus and urinary tract infections. To investigate the effect of Polygonum capitatum on cytochrome P450 (CYP) isoforms (CYP1A2, CYP2C9, CYP2C19, CYP2E1, and CYP3A4) in vivo using a "cocktail" approach by administering five probe drugs to rats. This study assessed the potential of Polygonum capitatum to interact with co-administered drugs.
机译:民族科医生相关性:Polygonum Capitatum是一个着名的苗族药用植物,这些植物已被用于对各种泌尿学疾病的独特治疗作用,包括泌尿微积分和泌尿道感染。 通过向大鼠施用五种探针药物,探讨体内细胞色素p450(CYP)同种型(CYP1A2,CYP2C9,CYP2C19,CYP2C19,CYP2C19,CYP2C19,CYP2C19,CYP2C19,CYP3A4)的影响。 该研究评估了助致的助致与共同施用的药物相互作用的潜力。

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  • 作者单位

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

    Guiyang Med Univ Sch Pharm Prov Key Lab Pharmaceut Guizhou Prov Guiyang 550004 Peoples R China;

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  • 原文格式 PDF
  • 正文语种 eng
  • 中图分类 药理学;
  • 关键词

    Polygonum capitatum; Cytochrome P450; Herb-drug interactions; Probe drug cocktail; UPLC-ESI-MS;

    机译:polygonum capitatum;细胞色素p450;草药相互作用;探针药物鸡尾酒;UPLC-ESI-MS;
  • 入库时间 2022-08-19 19:48:12

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