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机译:(R)-8-(6-甲基-4-氧代-1,4,5,6-四氢吡咯烷吡咯-2-基)-3-(1-甲基环丙基)-2- ((1-甲基环丙烯)氨基)喹唑啉-4(3H) - 血液恶性肿瘤的血液和选择性PIM-1/2激酶抑制剂
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Mol Struct One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Oncol Res One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Pharmacokinet &
Drug Metab One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Mol Struct One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Oncol Res One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Pharmacokinet &
Drug Metab One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Discovery Technol One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Mol Struct One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Oncol Res One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Oncol Res One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Mol Struct One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Discovery Technol One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Discovery Technol One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Oncol Res One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Oncol Res One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Discovery Technol One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Oncol Res One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Pharmaceut One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Pharmaceut One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Pharmacokinet &
Drug Metab One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Pharmacokinet &
Drug Metab One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
Amgen Res Dept Therareut Discovery Med Chem One Amgen Ctr Dr Thousand Oaks CA 91320 USA;
机译:(R)-8-(6-甲基-4-氧代-1,4,5,6-四氢吡咯烷吡咯-2-基)-3-(1-甲基环丙基)-2- ((1-甲基环丙烯)氨基)喹唑啉-4(3H) - 血液恶性肿瘤的血液和选择性PIM-1/2激酶抑制剂
机译:2-((3-氨基-4-甲基苯基)氨基)-N-(2-甲基-5-(3-(三氟甲基)苯甲酰胺基)苯基)-4-(甲基氨基)嘧啶-5-羧酰胺(CHMFL- ABL-053)作为慢性粒细胞白血病的有效,选择性和口服BCR-ABL / SRC / p38激酶抑制剂
机译:鉴定Ataxia Telanciectasia突变(ATM)激酶的有效,选择性和口服抑制剂:AZD0156的发现(8- {6- [3-(二甲基氨基)丙氧基] Pyridin-3-Y1} -3-甲基-1 - (四氢-2H-吡喃-4-基)-1,3-二氢-2H-咪唑[4,5-C]喹啉-2-一)
机译:N-(3-((2-甲氧基-4-((4-甲基-4-(4-甲基哌嗪-1-基)苯基)氨基)-4-甲基-2-氧代-2H-嘧啶的发现和生物学评价45 -d 13恶唑汀-1(4h) - 苯基)苯基)丙烯酰胺作为有效的Bruton的酪氨酸激酶抑制剂
机译:发现2((3-氨基-4-甲基苯基)氨基)N(2-甲基-5-(3-(三氟甲基)苯甲酰氨基)苯基)-4-(甲基氨基)嘧啶-5-甲酰胺(CHMFL-ABL-053 )作为慢性髓性白血病的有效,选择性和口服的BCR-ABL / SRC / P38激酶抑制剂