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机译:Braneburrinib(BMS-986195)的发现:一种识别高效和选择性共价抑制剂的策略,提供快速的Brution的酪氨酸激酶(BTK)的体内失活
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev POB 4000 Princeton NJ 08543 USA;
机译:Braneburrinib(BMS-986195)的发现:一种识别高效和选择性共价抑制剂的策略,提供快速的Brution的酪氨酸激酶(BTK)的体内失活
机译:发现丰富且具有高度选择性的Bruton酪氨酸激酶轴承三嗪脚手架的共价抑制剂
机译:LOU064(Rembribrutinib),富乐酪氨酸激酶的有效和高度选择性的共价抑制剂的发现
机译:CNX-774,Bruton的酪氨酸激酶的不可逆转,选择性和口服生物可利用的抑制剂:体外Adme,选择性和药代动力学性能
机译:靶向蛋白质酪氨酸激酶的RNAi筛选可将布鲁顿酪氨酸激酶(BTK)识别为乳腺癌细胞生存因子。
机译:发现高度有效和选择性的Bruton的酪氨酸激酶抑制剂避免了B细胞非霍奇金淋巴瘤的ADCC效应的损害
机译:伊布鲁替尼的发现:口服,有效和高度选择性,共价镇静的酪氨酸激酶(BTK)抑制剂用于治疗免疫疾病