...
机译:含有环氧酮的大环肽,具有口服可用性作为蛋白酶体抑制剂的致癌物质肽
Zhejiang Univ Coll Pharmaceut Sci ZJU ENS Joint Lab Med Chem Zhejiang Prov Key Lab Anti Canc Drug Res Hangzhou 310058 Zhejiang Peoples R China;
Chinese Acad Sci Natl Ctr Drug Screening Shanghai Inst Mat Med State Key Lab Drug Res Shanghai 201203 Peoples R China;
Anhui Univ Chinese Med Sch Pharm Dept Med Chem Hefei 230031 Anhui Peoples R China;
ShanghaiTech Univ Sch Life Sci &
Technol Shanghai 201203 Peoples R China;
Zhejiang Univ Coll Pharmaceut Sci ZJU ENS Joint Lab Med Chem Zhejiang Prov Key Lab Anti Canc Drug Res Hangzhou 310058 Zhejiang Peoples R China;
Chinese Acad Sci Natl Ctr Drug Screening Shanghai Inst Mat Med State Key Lab Drug Res Shanghai 201203 Peoples R China;
Chinese Acad Sci Natl Ctr Drug Screening Shanghai Inst Mat Med State Key Lab Drug Res Shanghai 201203 Peoples R China;
Zhejiang Univ City Coll Hangzhou 310015 Zhejiang Peoples R China;
Zhejiang Univ Coll Pharmaceut Sci ZJU ENS Joint Lab Med Chem Zhejiang Prov Key Lab Anti Canc Drug Res Hangzhou 310058 Zhejiang Peoples R China;
Chinese Acad Sci Natl Ctr Drug Screening Shanghai Inst Mat Med State Key Lab Drug Res Shanghai 201203 Peoples R China;
Zhejiang Univ Coll Pharmaceut Sci ZJU ENS Joint Lab Med Chem Zhejiang Prov Key Lab Anti Canc Drug Res Hangzhou 310058 Zhejiang Peoples R China;
Chinese Acad Sci Natl Ctr Drug Screening Shanghai Inst Mat Med State Key Lab Drug Res Shanghai 201203 Peoples R China;
Zhejiang Univ Coll Pharmaceut Sci ZJU ENS Joint Lab Med Chem Zhejiang Prov Key Lab Anti Canc Drug Res Hangzhou 310058 Zhejiang Peoples R China;
机译:含有环氧酮的大环肽,具有口服可用性作为蛋白酶体抑制剂的致癌物质肽
机译:新型具有环氧酮战斗部的蛋白酶体抑制剂的开发:非肽类贝拉糖酶衍生物与肽类环氧酮的合理杂交
机译:口服生物利用性和选择性肽环氧酮蛋白酶体抑制剂的设计与合成(PR-047)
机译:基于向日葵胰蛋白酶抑制剂-1的循环肽框架的开发口服可用素质蛋白
机译:蛋白质相互作用中大环肽抑制剂进化的策略
机译:从含尿素肽乙烯基砜的聚焦库中的有效且高度β1特异性蛋白酶体抑制剂的发现和肽环氧酮
机译:组合的3D-QSAR,分子对接和分子动力学研究肽环氧酮和酪肽素-硼酸作为抗人20S蛋白酶体β5亚基的抑制剂