MICROWAVE-ASSISTED CYCLOADDITION REACTION OF AZIDES TO N-SUBSTITUTED 2-AZABICYCLO[2.2.1]HEPT-5-EN-3-ONES

摘要

The reaction of N-substituted 2-azabicyclo[2.2.1]hept-5-en-3-ones (ABH)(1)with azides (2,4)could be effected under microwave conditions,producing aziridine-fused ABH (3)and triazolines (5,6)in good yields.