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Journal of enzyme inhibition

MEDLINE

中文名称：酶抑制杂志

ISSN：8755-5093
出版周期：6 no. a year

发文量：100

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1.Carbonic anhydrase inhibitors: synthesis of Schiff bases of hydroxybenzaldehydes with aromatic sulfonamides and their reactions with arylsulfonyl isocyanates.

机译：碳酸酐酶抑制剂：羟基苯甲醛Schiff碱与芳族磺酰胺的合成及其与芳基磺酰基异氰酸酯的反应。
- 作者：Scozzafava A;Banciu MD;Popescu A;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Carbonic Anhydrase Inhibitors;
- Benzaldehydes;
- Isocyanates;
- Schiff Bases;
- 碳酸酐酶抑制剂;
2.Use of a bisubstrate inhibitor to distinguish between isocitrate dehydrogenase isozymes.

机译：双底物抑制剂用于区分异柠檬酸脱氢酶同工酶的用途。
- 作者：Ehrlich RS
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
3.Carbonic anhydrase inhibitors; phosphoryl-sulfonamides--a new class of high affinity inhibitors of isozymes I and II.

机译：碳酸酐酶抑制剂;磷酰基磺酰胺-新型的同工酶I和II的高亲和力抑制剂。
- 作者：Fenesan I;Popescu R;Scozzafava A;Crucin V;Mateiciuc E;Bauer R;Ilies MA;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- Carbonate Dehydratase;
- Carbonic Anhydrase Inhibitors;
- Phosphoric Acid Esters;
- 碳酸脱水酶;
- 碳酸酐酶抑制剂;
- 磷酸酯类;
- 磺胺类;
4.A kinetic study on the interaction between tazobactam (a penicillanic acid sulphone derivative) and active-site serine beta-lactamases.

机译：他唑巴坦（青霉酸砜衍生物）与活性部位丝氨酸β-内酰胺酶相互作用的动力学研究。
- 作者：Perilli M;Franceschini N;Bonfiglio G;Segatore B;Stefani S;Nicoletti G;Perez MM;Bianchi C;Zollo A;Amicosante G
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Penicillanic Acid;
- Serine;
- beta-Lactamases;
- Enzyme Inhibitors;
- tazobactam;
- 青霉烷酸;
- 丝氨酸;
- β内酰胺酶类;
5.Alkaloidal sugar mimetics: biological activities and therapeutic applications.

机译：生物碱模拟糖：生物学活性和治疗应用。
- 作者：Asano N
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- Alkaloids;
- Carbohydrates;
- Glycoside Hydrolases;
- Molecular Mimicry;
- Hypoglycemic Agents;
- 生物碱类;
- 碳水化合物;
- 糖苷水解酶类;
- 分子模拟;
6.Carbonic anhydrase inhibitors: aromatic sulfonamides and disulfonamides act as efficient tumor growth inhibitors.

机译：碳酸酐酶抑制剂：芳族磺酰胺和二磺酰胺可作为有效的肿瘤生长抑制剂。
- 作者：Supuran CT io.chim.unifi.it;Scozzafava A
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Antineoplastic Agents;
- Carbonic Anhydrase Inhibitors;
- Arylsulfonates;
- Sulfonamides;
- 抗肿瘤药;
- 碳酸酐酶抑制剂;
7.Carbonic anhydrase activators: synthesis of high affinity isozymes I, II and IV activators, derivatives of 4-(arylsulfonylureido-amino acyl)ethyl-1H-imidazole.

机译：碳酸酐酶激活剂：高亲和力同工酶I，II和IV激活剂，4-（芳基磺酰基脲基-氨基酰基）乙基-1H-咪唑的衍生物。
- 作者：Supuran CT io.chim.unifi.it;Scozzafava A
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Carbonate Dehydratase;
- Enzyme Activators chemical synthesis;
- Imidazoles;
- 碳酸脱水酶;
- 咪唑类;
8.Carbonic anhydrase inhibitors. Synthesis of topically effective intraocular pressure lowering agents derived from 5-(omega-aminoalkylcarboxamido)-1,3,4-thiadiazole-2-sulfonamide.

机译：碳酸酐酶抑制剂。由5-（ω-氨基烷基羧酰胺基）-1,3,4-噻二唑-2-磺酰胺衍生的局部有效的眼内降压剂的合成。
- 作者：Barboiu M;Supuran CT;Menabuoni L;Scozzafava A;Mincione F;Briganti F;Mincione G
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Carbonic Anhydrase Inhibitors;
- Intraocular Pressure;
- Sulfonamides;
- Thiadiazoles;
- 碳酸酐酶抑制剂;
- 眼内压;
- 磺胺类;
- 噻二唑类;
9.Non-enzymatic glycosylation (or glycation) and inhibition of the pig heart cytosolic aspartate aminotransferase by glyceraldehyde 3-phosphate.

机译：非酶糖基化（或糖基化）和3-磷酸甘油醛对猪心脏胞质天冬氨酸转氨酶的抑制作用。
- 作者：Fitzgerald C;Swearengin TA;Yeargans G;McWhorter D;Cucchetti B;Seidler NW
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Aspartate Transaminase metabolism;
- Glyceraldehyde 3-Phosphate;
- Myocardium;
- 甘油醛3-磷酸酯;
- 心肌;
10.The kinetic mechanism of 5-enolpyruvylshikimate-3-phosphate synthase from a gram-positive pathogen Streptococcus pneumoniae.

机译：革兰氏阳性病原菌肺炎链球菌5-烯醇丙酮酸shi草酸酯-3-磷酸合酶的动力学机制。
- 作者：Du W;Wallis NG;Payne DJ
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Alkyl and Aryl Transferases;
- Glycine;
- Shikimic Acid;
- Streptococcus pneumoniae;
- 烷基和芳基转移酶类;
- 甘氨酸;
- 莽草酸;
- 链球菌;
- 肺炎;
11.Synthesis and mechanism of action of novel thiocarbamate inhibitors of human leukocyte elastase.

机译：人白细胞弹性蛋白酶的新型硫代氨基甲酸酯抑制剂的合成及其作用机理。
- 作者：Li-Pan ZS;Joshi HV;Digenis GA
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
12.Influence of stereoisomers of 4-fluoroglutamate on rat brain glutamate decarboxylase.

机译：4-氟谷氨酸的立体异构体对大鼠脑谷氨酸脱羧酶的影响。
- 作者：Drsata J;Netopilova M;Tolman V
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- Brain;
- Glutamate Decarboxylase;
- Glutamates;
- Enzyme Inhibitors;
- 4-fluoroglutamic acid;
- 脑;
- 谷氨酸脱羧酶;
- 谷氨酸盐类;
13.Dye affinity labelling of yeast alcohol dehydrogenase.

机译：酵母酒精脱氢酶的染料亲和标记。
- 作者：Labrou NE;uadec.aua.gr
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Affinity Labels;
- Alcohol Dehydrogenase;
- Anthraquinones;
- Dyes;
- Saccharomyces;
- 亲和力标记物;
- 醇脱氢酶;
- 蒽醌类;
- 染料;
- 酵母菌属;
- 三嗪类;
14.Glucosylated isoflavones as DNA topoisomerase II poisons.

机译：糖基化异黄酮是DNA拓扑异构酶II的毒物。
- 作者：Martin-Cordero C;Lopez-Lazaro M;Pinero J;Ortiz T;Cortes F;Ayuso MJ
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- DNA Topoisomerase ATP Hydrolysing antagonists and inhibitors;
- Drugs;
- Chinese Herbal;
- 中草药;
- 酶抑制剂;
- 雌激素类;
- 非甾类;
- 异黄酮类;
15.Expression in yeast and purification of functional recombinant human poly(ADP-ribose)polymerase (PARP). Comparative pharmacological profile with that of the rat enzyme.

机译：在酵母中表达和功能重组人聚（ADP-核糖）聚合酶（PARP）的纯化。与大鼠酶比较的药理特性。
- 作者：Perrin D;Gras S;van-Hille B;Hill BT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- 1-Naphthylamine;
- Enzyme Inhibitors;
- NAD+ ADP-Ribosyltransferase;
- Saccharomyces;
- 1-萘胺;
- 酶抑制剂;
- NAD+ADP核糖转移酶;
- 酵母菌属;
- 睾丸;
16.Antifungal activity of Ag(I) and Zn(II) complexes of aminobenzolamide (5-sulfanilylamido-1,3,4-thiadiazole-2-sulfonamide) derivatives.

机译：氨基苯甲酰胺（5-磺胺基酰胺基-1,3,4-噻二唑-2-磺酰胺）衍生物的Ag（I）和Zn（II）配合物的抗真菌活性。
- 作者：Mastrolorenzo A;Scozzafava A;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Antifungal Agents;
- Carbonic Anhydrase Inhibitors;
- Sulfonamides;
- Aminobenzoic Acids;
- 抗真菌药;
- 碳酸酐酶抑制剂;
- 磺胺类;
17.Inhibition of AChE: structure-activity relationship among conformational transition of Trp84 and biomolecular rate constant.

机译：抑制AChE：Trp84构象转变与生物分子速率常数之间的构效关系。
- 作者：Bertonati C;Marta M;Patamia M;Colella A;Pomponi M
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Acetylcholinesterase;
- Carbamates;
- Cholinesterase Inhibitors;
- 乙酰胆碱酯酶;
- 氨甲酸酯类;
- 胆碱酯酶抑制剂;
18.Selective inhibition of monoamine oxidase B by aminoethyl substituted benzyl ethers.

机译：氨乙基取代的苄基醚对单胺氧化酶B的选择性抑制。
- 作者：Woodroofe CC;Mostashari R;Lu X;Ramsay RR;Silverman RB
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Benzyl Compounds;
- Isoenzymes;
- Monoamine Oxidase;
- Monoamine Oxidase Inhibitors;
- 苄基化合物;
- 同工酶类;
- 单胺氧化酶;
- 单胺氧化酶抑制剂;
19.Inhibition of glutathione reductase by isoproterenol oxidation products.

机译：异丙肾上腺素氧化产物对谷胱甘肽还原酶的抑制作用。
- 作者：Remiao F;Carmo H;Carvalho FD;Bastos ML
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Glutathione Reductase;
- Isoproterenol;
- Antioxidants;
- Indicators and Reagents;
- 谷胱甘肽还原酶;
- 异丙肾上腺素;
20.Competitive inhibition of Trypanosoma brucei phosphoglucose isomerase by D-arabinose-5-phosphate derivatives.

机译：D-阿拉伯糖-5-磷酸酯衍生物竞争抑制布鲁氏锥虫磷酸葡萄糖异构酶。
- 作者：Hardre R;Salmon L;Opperdoes FR
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Enzyme Inhibitors;
- Glucose 6 Phosphate Isomerase antagonists and inhibitors;
- 酶抑制剂;
- 戊糖磷酸类;
- 锥虫;
- 布鲁斯布鲁斯;
21.The antifungal activity of sulfonylated/carboxylated derivatives of dibenzo-1,4-dioxine-2-acetyloxime may be due to inhibition of lanosterol-14alpha-demethylase.

机译：二苯并-1,4-二恶英-2-乙酰肟的磺化/羧化衍生物的抗真菌活性可能是由于抑制了羊毛甾醇-14α-脱甲基酶。
- 作者：Mastrolorenzo A;Scozzafava A;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Antifungal Agents;
- Carbamates;
- Cytochrome P-450;
- Oxidoreductases;
- Alkanesulfonates;
- 抗真菌药;
- 氨甲酸酯类;
- 细胞色素P-450;
- 氧化还原酶类;
22.Inhibition of rabbit muscle isozymes by vitamin C.

机译：维生素C对兔肌肉同工酶的抑制作用
- 作者：Russell PJ;Williams A;Austin TA
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- 6-Phosphofructokinase;
- Adenylate Kinase;
- Ascorbic Acid;
- Lactate Dehydrogenase;
- 6-磷酸果糖激酶;
- 腺苷酸激酶;
- 抗坏血酸;
- 乳酸脱氢酶;
- 肌;
- 骨骼;
23.Protease inhibitors. Part 2. Weakly basic thrombin inhibitors incorporating sulfonyl-aminoguanidine moieties as S1 anchoring groups: synthesis and structure-activity correlations.

机译：蛋白酶抑制剂。第2部分。弱碱性凝血酶抑制剂，将磺酰基-氨基胍部分作为S1锚定基团：合成与结构活性相关。
- 作者：Clare BW;Scozzafava A;Briganti F;Iorga B;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- Antithrombins;
- Guanidines;
- Serine Proteinase Inhibitors;
- Sulfones;
- Thrombin;
- 抗凝血酶类;
- 胍类;
- 丝氨酸蛋白酶抑制剂;
- 砜类;
- 凝血酶;
24.Interaction of pig kidney and lentil seedling copper-containing amine oxidases with guanidinium compounds.

机译：猪肾和扁豆幼苗含铜胺氧化酶与胍盐化合物的相互作用。
- 作者：Padiglia A;Medda R;Lorrai A;Murgia B;Pedersen JZ;Agro AF;Floris G
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
25.N3-oxoacyl derivatives of L-2,3-diaminopropanoic acid and their peptides; novel inhibitors of glucosamine-6-phosphate synthase.

机译：L-2，3-二氨基丙酸的N3-氧酰基衍生物及其肽;氨基葡萄糖6-磷酸合酶的新型抑制剂。
- 作者：Andruszkiewicz R;Jedrzejczak R;Zieniawa T;Wojciechowski M;Borowski E
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
26.Carbonic anhydrase inhibitors: inhibition of isozymes I, II and IV by sulfamide and sulfamic acid derivatives.

机译：碳酸酐酶抑制剂：磺酰胺和氨基磺酸衍生物抑制同工酶I，II和IV。
- 作者：Scozzafava A;Banciu MD;Popescu A;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Carbonate Dehydratase;
- Carbonic Anhydrase Inhibitors;
- Sulfonamides;
- Sulfonic Acids;
- 碳酸脱水酶;
- 碳酸酐酶抑制剂;
- 磺胺类;
- 磺酸类;
27.Nickel-induced substrate inhibition of bovine liver glutamate dehydrogenase.

机译：镍诱导的牛肝谷氨酸脱氢酶的底物抑制。
- 作者：Ghobadi S;Nemat-Gorgani M;Golabi SM;Zare HR;Moosavi-Movahedi AA
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Glutamate Dehydrogenase;
- Liver;
- NAD;
- Nickel;
- Ketoglutaric Acids;
- Ammonia;
- 谷氨酸脱氢酶;
- 肝;
- 镍;
28.Invertase proteinaceous inhibitor of Cyphomandra betacea Sendt fruits.

机译：拟南芥甜菜果实的转化酶蛋白抑制剂。
- 作者：Ordonez RM;Isla MI;Vattuone MA;Sampietro AR
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Fruit;
- Glycoside Hydrolases;
- Enzyme Inhibitors;
- Lectins;
- Plant Proteins;
- 水果;
- 糖苷水解酶类;
29.Non-linear slow-binding inhibition of Aerococcus viridans lactate oxidase by Cibacron Blue 3GA.

机译：Cibacron Blue 3GA对绿球菌乳酸氧化酶的非线性慢结合抑制。
- 作者：Streitenberger-S A;Lopez-Mas-J A;Sanchez-Ferrer A;Garcia-Carmona F
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Blue color;
- binding;
- Psychological inhibition;
- Slow;
- Gaffkya homari;
30.Enantioselectivity of some 1-((benzofuran-2-yl) phenylmethyl) imidazoles as aromatase (P450AROM) inhibitors.

机译：一些1-（（（苯并呋喃-2-基）苯基甲基）咪唑作为芳香酶（P450AROM）抑制剂的对映选择性。
- 作者：Khodarahmi-G A;Laughton-C A;Smith-H J;Nicholls-P J
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第5期
- Upper case ess;
- Joule;
- Unit of energy;
- inhibitors;
- Carbon ion;
- benzofuran;
31.Inhibition of potato polyphenol oxidase by anions and activity in various carboxylate buffers (pH 4.8) at constant ionic strength.

机译：在恒定的离子强度下，阴离子对马铃薯多酚氧化酶的抑制作用和在各种羧酸盐缓冲液（pH 4.8）中的活性。
- 作者：Malkin BD;Thickman KR;Markworth CJ;Wilcox DE;Kull FJ
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第2期
- Carboxylic Acids;
- Catechol Oxidase;
- Enzyme Inhibitors;
- Potatoes;
- Buffers;
- 羧酸类;
- 儿茶酚氧化酶;
- 酶抑制剂;
- 马铃薯;
32.Quantitative structure-activity relationship of some HIV-1 protease inhibitors: a Fujita-Ban type analysis.

机译：某些HIV-1蛋白酶抑制剂的定量构效关系：Fujita-Ban类型分析。
- 作者：Mekapati SB;Sivakumar R;Gupta SP
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- Analysis of substances;
- Physical activity;
33.Allosteric inhibition of rat liver and kidney arginase by copper and mercury ions.

机译：铜和汞离子对大鼠肝脏和肾脏精氨酸酶的变构抑制作用。
- 作者：Tormanen-C D
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第5期
- Arginase;
- Psychological inhibition;
- Isoenzymes;
- Liver;
- Kidney;
- 精氨酸酶;
- 同工酶类;
- 肝;
- 肾;
34.Effects of substrate structural analogues on the enzymatic activities of aspartate aminotransferase isoenzymes.

机译：底物结构类似物对天冬氨酸转氨酶同工酶的酶活性的影响。
- 作者：Martins LL;Mourato MP;de-Varennes A
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- alpha 1-Antitrypsin;
- Donors;
- Isoenzymes;
- -4;
- α1-抗胰蛋白酶;
- 同工酶类;
35.Purification and characterization of catalase from chard (Beta vulgaris var. cicla).

机译：唐莴苣（Beta vulgaris var。cicla）中过氧化氢酶的纯化和鉴定。
- 作者：Dincer A;Aydemir T
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第2期
- Catalase;
- Chenopodiaceae;
- Chlorides;
- Enzyme Inhibitors;
- Ferric Compounds;
- 过氧化氢酶;
- 藜科;
36.Glycosylasparaginase inhibition studies: competitive inhibitors, transition state mimics, noncompetitive inhibitors.

机译：糖基葡聚糖酶抑制研究：竞争性抑制剂，过渡态模拟物，非竞争性抑制剂。
- 作者：Risley JM;Huang DH;Kaylor JJ;Malik JJ;Xia YQ
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- Aspartylglucosylaminase;
- competition;
- inhibitors;
- VALUING;
- 天冬氨酰葡糖脱氨基酶;
37.Quantitative structure-activity relationship study of novel alpha1a-selective adrenoceptor antagonists.

机译：新型α1a-选择性肾上腺素受体拮抗剂的定量构效关系研究。
- 作者：Singh P;Kumar R
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- structure;
- antagonists;
- novel;
- KAI1 Gene;
- Upper case ecks;
38.Quantitative structure-activity relationships (QSARs) within series of inhibitors for mammalian cytochromes P450 (CYPs).

机译：哺乳动物细胞色素P450（CYPs）抑制剂系列中的定量构效关系（QSAR）。
- 作者：Lewis-D F;Dickins M
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Quantitative Structure-Activity Relationship;
- structure;
- inhibitors;
- lipophilicity;
39.Inhibition of pig liver and Zea mays L. polyamine oxidase: a comparative study.

机译：猪肝和玉米玉米多胺氧化酶的抑制作用：一项比较研究。
- 作者：Federico R;Leone L;Botta M;Binda C;Angelini R;Venturini G;Ascenzi P
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第2期
- Amine Oxidoreductases;
- Corn;
- Enzyme Inhibitors;
- Liver;
- Benzamidines;
- Guanidines;
- 胺氧化还原酶类;
- 玉米;
- 酶抑制剂;
- 肝;
40.Kinetics of inactivation of Ulva pertusa Kjellm alkaline phosphatase by ethylenediaminetetraacetic acid disodium.

机译：乙二胺四乙酸二钠灭活百日草碱性磷酸酶的动力学。
- 作者：Yang D;Wang J;Peng X;An L
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Edetic Acid;
- Ulva;
- kinetic characteristics;
- Enzymes;
- Alkaline Phosphatase;
- 依地酸;
- 酶类;
- 碱性磷酸酶;
41.Isomerase activity of the C-terminal fructose-6-phosphate binding domain of glucosamine-6-phosphate synthase from Escherichia coli.

机译：大肠杆菌的氨基葡萄糖-6-磷酸合酶的C-末端果糖6-磷酸结合域的异构酶活性。
- 作者：Todorova R
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- binding;
- Carbon ion;
- inorganic phosphate;
- Isomerases;
- Glucosamine;
- 异构酶类;
- 葡糖胺;
42.Inhibition of Saccharomyces cerevisiae phosphomannose isomerase by the NO-donor S-nitroso-acetyl-penicillamine.

机译：NO供体S-亚硝基-乙酰基-青霉胺对酿酒酵母磷酸甘露糖异构酶的抑制作用。
- 作者：Salvati L;Mattu M;Tiberi F;Polticelli F;Ascenzi P
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- Saccharomyces cerevisiae;
- Mannose-6-Phosphate Isomerase;
- Donors;
- Penicillamine;
- 酵母菌;
- 酿酒;
- 青霉胺;
43.Evidence for an essential arginine in the flavoprotein nitroalkane oxidase.

机译：黄素蛋白硝基烷氧化酶中必需精氨酸的证据。
- 作者：Gadda G;Banerjee A;Fleming GS;Fitzpatrick PF
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第2期
- Arginine;
- Enzyme Inhibitors;
- Flavoproteins;
- Fusarium;
- Oxygenases;
- Cyclohexanones;
- 精氨酸;
- 酶抑制剂;
- 黄素蛋白类;
- 镰刀菌属;
- 氧合酶类;
44.A new class of potent reversible inhibitors of metallo-proteinases: C-terminal thiol-peptides as zinc-coordinating ligands.

机译：一类新的有效的金属蛋白酶可逆抑制剂：C末端硫醇肽作为锌配位体。
- 作者：Peters K;Jahreis G;Kotters-E M
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Peptides;
- inhibitors;
- Sulfhydryl Compounds;
- Zinc;
- Carbon ion;
- 肽类;
- 巯基化合物;
- 锌;
45.Synthesis and evaluation of dipeptide amides containing N omega-nitroarginine and D-2,4-diaminobutyric acids as inhibitors of neuronal nitric oxide synthase.

机译：包含Nω-硝基精氨酸和D-2,4-二氨基丁酸作为神经元一氧化氮合酶抑制剂的二肽酰胺的合成和评估。
- 作者：Huang H;Martasek P;Roman LJ;Silverman RB
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- Dipeptides;
- Amides;
- Containing;
- inhibitors;
- Neuronal;
- Nitric-Oxide Synthase;
- 二肽类;
- 酰胺类;
- 一氧化氮合酶;
- 氮芥;
46.Structure-activity relationships of new NAPAP-analogs.

机译：新的NAPAP模拟物的构效关系。
- 作者：Steinmetzer T;Schweinitz A;Kunzel S;Wikstrom P;Hauptmann J;Sturzebecher J
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- New;
- analogs;
- Thrombin;
- 凝血酶;
47.Carbonic anhydrase activity modulators: synthesis of inhibitors and activators incorporating 2-substituted-thiazol-4-yl-methyl scaffolds.

机译：碳酸酐酶活性调节剂：结合了2-取代的噻唑-4-基甲基支架的抑制剂和活化剂的合成。
- 作者：Scozzafava A;Saramet I;Banciu-M D;Supuran-C T
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- AC protocol;
- inhibitors;
- Carbonic Anhydrases;
- Roman Numeral IV;
- sulfamate;
48.Progress curves analysis as an alternative for exploration of activation-inhibition phenomena in cholinesterases.

机译：进度曲线分析可作为探索胆碱酯酶激活抑制现象的替代方法。
- 作者：Golicnik M
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第5期
- Analysis of substances;
- Psychological inhibition;
- Acetylcholinesterase;
- agreement;
- 乙酰胆碱酯酶;
49.Inhibition of succinate-cytochrome C reductase by a ferromacrocyclic complex.

机译：亚铁大环复合物抑制琥珀酸-细胞色素C还原酶。
- 作者：Balbaa M;Khalifa M;el-Sabawaya M;Kandeel K
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Psychological inhibition;
- Enzymes;
- Lower case sea;
- succinate;
- Cytochrome c;
- 酶类;
- 细胞色素C;
50.A 3D QSAR study of monoamino oxidase-B inhibitors using the chemical function based pharmacophore generation approach.

机译：使用基于化学功能的药效团产生方法对单氨基氧化酶-B抑制剂进行3D QSAR研究。
- 作者：Gritsch S;Guccione S;Hoffmann R;Cambria A;Raciti G;Langer T
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- inhibitors;
- Chemical compound;
- NOS;
- pharmacophore;
- Type B Monoamine Oxidase;
51.Carbonic anhydrase inhibitors: synthesis of Schiff bases of hydroxybenzaldehydes with aromatic sulfonamides and their reactions with arylsulfonyl isocyanates.

机译：碳酸酐酶抑制剂：羟基苯甲醛Schiff碱与芳族磺酰胺的合成及其与芳基磺酰基异氰酸酯的反应。
- 作者：Scozzafava A;Banciu MD;Popescu A;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Carbonic Anhydrase Inhibitors;
- Benzaldehydes;
- Isocyanates;
- Schiff Bases;
- 碳酸酐酶抑制剂;
52.Carbonic anhydrase inhibitors; phosphoryl-sulfonamides--a new class of high affinity inhibitors of isozymes I and II.

机译：碳酸酐酶抑制剂;磷酰基磺酰胺-新型的同工酶I和II的高亲和力抑制剂。
- 作者：Fenesan I;Popescu R;Scozzafava A;Crucin V;Mateiciuc E;Bauer R;Ilies MA;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- Carbonate Dehydratase;
- Carbonic Anhydrase Inhibitors;
- Phosphoric Acid Esters;
- 碳酸脱水酶;
- 碳酸酐酶抑制剂;
- 磷酸酯类;
- 磺胺类;
53.Use of a bisubstrate inhibitor to distinguish between isocitrate dehydrogenase isozymes.

机译：双底物抑制剂用于区分异柠檬酸脱氢酶同工酶的用途。
- 作者：Ehrlich RS
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
54.A kinetic study on the interaction between tazobactam (a penicillanic acid sulphone derivative) and active-site serine beta-lactamases.

机译：他唑巴坦（青霉酸砜衍生物）与活性部位丝氨酸β-内酰胺酶相互作用的动力学研究。
- 作者：Perilli M;Franceschini N;Bonfiglio G;Segatore B;Stefani S;Nicoletti G;Perez MM;Bianchi C;Zollo A;Amicosante G
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Penicillanic Acid;
- Serine;
- beta-Lactamases;
- Enzyme Inhibitors;
- tazobactam;
- 青霉烷酸;
- 丝氨酸;
- β内酰胺酶类;
55.Carbonic anhydrase inhibitors: aromatic sulfonamides and disulfonamides act as efficient tumor growth inhibitors.

机译：碳酸酐酶抑制剂：芳族磺酰胺和二磺酰胺可作为有效的肿瘤生长抑制剂。
- 作者：Supuran CT io.chim.unifi.it;Scozzafava A
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Antineoplastic Agents;
- Carbonic Anhydrase Inhibitors;
- Arylsulfonates;
- Sulfonamides;
- 抗肿瘤药;
- 碳酸酐酶抑制剂;
56.Alkaloidal sugar mimetics: biological activities and therapeutic applications.

机译：生物碱模拟糖：生物学活性和治疗应用。
- 作者：Asano N
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- Alkaloids;
- Carbohydrates;
- Glycoside Hydrolases;
- Molecular Mimicry;
- Hypoglycemic Agents;
- 生物碱类;
- 碳水化合物;
- 糖苷水解酶类;
- 分子模拟;
57.Carbonic anhydrase activators: synthesis of high affinity isozymes I, II and IV activators, derivatives of 4-(arylsulfonylureido-amino acyl)ethyl-1H-imidazole.

机译：碳酸酐酶激活剂：高亲和力同工酶I，II和IV激活剂，4-（芳基磺酰基脲基-氨基酰基）乙基-1H-咪唑的衍生物。
- 作者：Supuran CT io.chim.unifi.it;Scozzafava A
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Carbonate Dehydratase;
- Enzyme Activators chemical synthesis;
- Imidazoles;
- 碳酸脱水酶;
- 咪唑类;
58.Carbonic anhydrase inhibitors. Synthesis of topically effective intraocular pressure lowering agents derived from 5-(omega-aminoalkylcarboxamido)-1,3,4-thiadiazole-2-sulfonamide.

机译：碳酸酐酶抑制剂。由5-（ω-氨基烷基羧酰胺基）-1,3,4-噻二唑-2-磺酰胺衍生的局部有效的眼内降压剂的合成。
- 作者：Barboiu M;Supuran CT;Menabuoni L;Scozzafava A;Mincione F;Briganti F;Mincione G
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Carbonic Anhydrase Inhibitors;
- Intraocular Pressure;
- Sulfonamides;
- Thiadiazoles;
- 碳酸酐酶抑制剂;
- 眼内压;
- 磺胺类;
- 噻二唑类;
59.Non-enzymatic glycosylation (or glycation) and inhibition of the pig heart cytosolic aspartate aminotransferase by glyceraldehyde 3-phosphate.

机译：非酶糖基化（或糖基化）和3-磷酸甘油醛对猪心脏胞质天冬氨酸转氨酶的抑制作用。
- 作者：Fitzgerald C;Swearengin TA;Yeargans G;McWhorter D;Cucchetti B;Seidler NW
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Aspartate Transaminase metabolism;
- Glyceraldehyde 3-Phosphate;
- Myocardium;
- 甘油醛3-磷酸酯;
- 心肌;
60.Synthesis and mechanism of action of novel thiocarbamate inhibitors of human leukocyte elastase.

机译：人白细胞弹性蛋白酶的新型硫代氨基甲酸酯抑制剂的合成及其作用机理。
- 作者：Li-Pan ZS;Joshi HV;Digenis GA
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
61.The kinetic mechanism of 5-enolpyruvylshikimate-3-phosphate synthase from a gram-positive pathogen Streptococcus pneumoniae.

机译：革兰氏阳性病原菌肺炎链球菌5-烯醇丙酮酸shi草酸酯-3-磷酸合酶的动力学机制。
- 作者：Du W;Wallis NG;Payne DJ
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Alkyl and Aryl Transferases;
- Glycine;
- Shikimic Acid;
- Streptococcus pneumoniae;
- 烷基和芳基转移酶类;
- 甘氨酸;
- 莽草酸;
- 链球菌;
- 肺炎;
62.Influence of stereoisomers of 4-fluoroglutamate on rat brain glutamate decarboxylase.

机译：4-氟谷氨酸的立体异构体对大鼠脑谷氨酸脱羧酶的影响。
- 作者：Drsata J;Netopilova M;Tolman V
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- Brain;
- Glutamate Decarboxylase;
- Glutamates;
- Enzyme Inhibitors;
- 4-fluoroglutamic acid;
- 脑;
- 谷氨酸脱羧酶;
- 谷氨酸盐类;
63.Dye affinity labelling of yeast alcohol dehydrogenase.

机译：酵母酒精脱氢酶的染料亲和标记。
- 作者：Labrou NE;uadec.aua.gr
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Affinity Labels;
- Alcohol Dehydrogenase;
- Anthraquinones;
- Dyes;
- Saccharomyces;
- 亲和力标记物;
- 醇脱氢酶;
- 蒽醌类;
- 染料;
- 酵母菌属;
- 三嗪类;
64.Glucosylated isoflavones as DNA topoisomerase II poisons.

机译：糖基化异黄酮是DNA拓扑异构酶II的毒物。
- 作者：Martin-Cordero C;Lopez-Lazaro M;Pinero J;Ortiz T;Cortes F;Ayuso MJ
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- DNA Topoisomerase ATP Hydrolysing antagonists and inhibitors;
- Drugs;
- Chinese Herbal;
- 中草药;
- 酶抑制剂;
- 雌激素类;
- 非甾类;
- 异黄酮类;
65.Expression in yeast and purification of functional recombinant human poly(ADP-ribose)polymerase (PARP). Comparative pharmacological profile with that of the rat enzyme.

机译：在酵母中表达和功能重组人聚（ADP-核糖）聚合酶（PARP）的纯化。与大鼠酶比较的药理特性。
- 作者：Perrin D;Gras S;van-Hille B;Hill BT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- 1-Naphthylamine;
- Enzyme Inhibitors;
- NAD+ ADP-Ribosyltransferase;
- Saccharomyces;
- 1-萘胺;
- 酶抑制剂;
- NAD+ADP核糖转移酶;
- 酵母菌属;
- 睾丸;
66.Antifungal activity of Ag(I) and Zn(II) complexes of aminobenzolamide (5-sulfanilylamido-1,3,4-thiadiazole-2-sulfonamide) derivatives.

机译：氨基苯甲酰胺（5-磺胺基酰胺基-1,3,4-噻二唑-2-磺酰胺）衍生物的Ag（I）和Zn（II）配合物的抗真菌活性。
- 作者：Mastrolorenzo A;Scozzafava A;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Antifungal Agents;
- Carbonic Anhydrase Inhibitors;
- Sulfonamides;
- Aminobenzoic Acids;
- 抗真菌药;
- 碳酸酐酶抑制剂;
- 磺胺类;
67.Inhibition of AChE: structure-activity relationship among conformational transition of Trp84 and biomolecular rate constant.

机译：抑制AChE：Trp84构象转变与生物分子速率常数之间的构效关系。
- 作者：Bertonati C;Marta M;Patamia M;Colella A;Pomponi M
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Acetylcholinesterase;
- Carbamates;
- Cholinesterase Inhibitors;
- 乙酰胆碱酯酶;
- 氨甲酸酯类;
- 胆碱酯酶抑制剂;
68.Selective inhibition of monoamine oxidase B by aminoethyl substituted benzyl ethers.

机译：氨乙基取代的苄基醚对单胺氧化酶B的选择性抑制。
- 作者：Woodroofe CC;Mostashari R;Lu X;Ramsay RR;Silverman RB
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Benzyl Compounds;
- Isoenzymes;
- Monoamine Oxidase;
- Monoamine Oxidase Inhibitors;
- 苄基化合物;
- 同工酶类;
- 单胺氧化酶;
- 单胺氧化酶抑制剂;
69.Inhibition of glutathione reductase by isoproterenol oxidation products.

机译：异丙肾上腺素氧化产物对谷胱甘肽还原酶的抑制作用。
- 作者：Remiao F;Carmo H;Carvalho FD;Bastos ML
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
- Glutathione Reductase;
- Isoproterenol;
- Antioxidants;
- Indicators and Reagents;
- 谷胱甘肽还原酶;
- 异丙肾上腺素;
70.Inhibition of rabbit muscle isozymes by vitamin C.

机译：维生素C对兔肌肉同工酶的抑制作用
- 作者：Russell PJ;Williams A;Austin TA
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- 6-Phosphofructokinase;
- Adenylate Kinase;
- Ascorbic Acid;
- Lactate Dehydrogenase;
- 6-磷酸果糖激酶;
- 腺苷酸激酶;
- 抗坏血酸;
- 乳酸脱氢酶;
- 肌;
- 骨骼;
71.Competitive inhibition of Trypanosoma brucei phosphoglucose isomerase by D-arabinose-5-phosphate derivatives.

机译：D-阿拉伯糖-5-磷酸酯衍生物竞争抑制布鲁氏锥虫磷酸葡萄糖异构酶。
- 作者：Hardre R;Salmon L;Opperdoes FR
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Enzyme Inhibitors;
- Glucose 6 Phosphate Isomerase antagonists and inhibitors;
- 酶抑制剂;
- 戊糖磷酸类;
- 锥虫;
- 布鲁斯布鲁斯;
72.The antifungal activity of sulfonylated/carboxylated derivatives of dibenzo-1,4-dioxine-2-acetyloxime may be due to inhibition of lanosterol-14alpha-demethylase.

机译：二苯并-1,4-二恶英-2-乙酰肟的磺化/羧化衍生物的抗真菌活性可能是由于抑制了羊毛甾醇-14α-脱甲基酶。
- 作者：Mastrolorenzo A;Scozzafava A;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Antifungal Agents;
- Carbamates;
- Cytochrome P-450;
- Oxidoreductases;
- Alkanesulfonates;
- 抗真菌药;
- 氨甲酸酯类;
- 细胞色素P-450;
- 氧化还原酶类;
73.Protease inhibitors. Part 2. Weakly basic thrombin inhibitors incorporating sulfonyl-aminoguanidine moieties as S1 anchoring groups: synthesis and structure-activity correlations.

机译：蛋白酶抑制剂。第2部分。弱碱性凝血酶抑制剂，将磺酰基-氨基胍部分作为S1锚定基团：合成与结构活性相关。
- 作者：Clare BW;Scozzafava A;Briganti F;Iorga B;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第3期
- Antithrombins;
- Guanidines;
- Serine Proteinase Inhibitors;
- Sulfones;
- Thrombin;
- 抗凝血酶类;
- 胍类;
- 丝氨酸蛋白酶抑制剂;
- 砜类;
- 凝血酶;
74.N3-oxoacyl derivatives of L-2,3-diaminopropanoic acid and their peptides; novel inhibitors of glucosamine-6-phosphate synthase.

机译：L-2，3-二氨基丙酸的N3-氧酰基衍生物及其肽;氨基葡萄糖6-磷酸合酶的新型抑制剂。
- 作者：Andruszkiewicz R;Jedrzejczak R;Zieniawa T;Wojciechowski M;Borowski E
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
75.Interaction of pig kidney and lentil seedling copper-containing amine oxidases with guanidinium compounds.

机译：猪肾和扁豆幼苗含铜胺氧化酶与胍盐化合物的相互作用。
- 作者：Padiglia A;Medda R;Lorrai A;Murgia B;Pedersen JZ;Agro AF;Floris G
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第1期
76.Nickel-induced substrate inhibition of bovine liver glutamate dehydrogenase.

机译：镍诱导的牛肝谷氨酸脱氢酶的底物抑制。
- 作者：Ghobadi S;Nemat-Gorgani M;Golabi SM;Zare HR;Moosavi-Movahedi AA
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Glutamate Dehydrogenase;
- Liver;
- NAD;
- Nickel;
- Ketoglutaric Acids;
- Ammonia;
- 谷氨酸脱氢酶;
- 肝;
- 镍;
77.Carbonic anhydrase inhibitors: inhibition of isozymes I, II and IV by sulfamide and sulfamic acid derivatives.

机译：碳酸酐酶抑制剂：磺酰胺和氨基磺酸衍生物抑制同工酶I，II和IV。
- 作者：Scozzafava A;Banciu MD;Popescu A;Supuran CT
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第5期
- Carbonate Dehydratase;
- Carbonic Anhydrase Inhibitors;
- Sulfonamides;
- Sulfonic Acids;
- 碳酸脱水酶;
- 碳酸酐酶抑制剂;
- 磺胺类;
- 磺酸类;
78.Invertase proteinaceous inhibitor of Cyphomandra betacea Sendt fruits.

机译：拟南芥甜菜果实的转化酶蛋白抑制剂。
- 作者：Ordonez RM;Isla MI;Vattuone MA;Sampietro AR
- 期刊名称：《Journal of enzyme inhibition》 | 2000年第6期
- Fruit;
- Glycoside Hydrolases;
- Enzyme Inhibitors;
- Lectins;
- Plant Proteins;
- 水果;
- 糖苷水解酶类;
79.Inhibition of potato polyphenol oxidase by anions and activity in various carboxylate buffers (pH 4.8) at constant ionic strength.

机译：在恒定的离子强度下，阴离子对马铃薯多酚氧化酶的抑制作用和在各种羧酸盐缓冲液（pH 4.8）中的活性。
- 作者：Malkin BD;Thickman KR;Markworth CJ;Wilcox DE;Kull FJ
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第2期
- Carboxylic Acids;
- Catechol Oxidase;
- Enzyme Inhibitors;
- Potatoes;
- Buffers;
- 羧酸类;
- 儿茶酚氧化酶;
- 酶抑制剂;
- 马铃薯;
80.Quantitative structure-activity relationship of some HIV-1 protease inhibitors: a Fujita-Ban type analysis.

机译：某些HIV-1蛋白酶抑制剂的定量构效关系：Fujita-Ban类型分析。
- 作者：Mekapati SB;Sivakumar R;Gupta SP
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- Analysis of substances;
- Physical activity;
81.Enantioselectivity of some 1-((benzofuran-2-yl) phenylmethyl) imidazoles as aromatase (P450AROM) inhibitors.

机译：一些1-（（（苯并呋喃-2-基）苯基甲基）咪唑作为芳香酶（P450AROM）抑制剂的对映选择性。
- 作者：Khodarahmi-G A;Laughton-C A;Smith-H J;Nicholls-P J
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第5期
- Upper case ess;
- Joule;
- Unit of energy;
- inhibitors;
- Carbon ion;
- benzofuran;
82.Non-linear slow-binding inhibition of Aerococcus viridans lactate oxidase by Cibacron Blue 3GA.

机译：Cibacron Blue 3GA对绿球菌乳酸氧化酶的非线性慢结合抑制。
- 作者：Streitenberger-S A;Lopez-Mas-J A;Sanchez-Ferrer A;Garcia-Carmona F
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Blue color;
- binding;
- Psychological inhibition;
- Slow;
- Gaffkya homari;
83.Allosteric inhibition of rat liver and kidney arginase by copper and mercury ions.

机译：铜和汞离子对大鼠肝脏和肾脏精氨酸酶的变构抑制作用。
- 作者：Tormanen-C D
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第5期
- Arginase;
- Psychological inhibition;
- Isoenzymes;
- Liver;
- Kidney;
- 精氨酸酶;
- 同工酶类;
- 肝;
- 肾;
84.Purification and characterization of catalase from chard (Beta vulgaris var. cicla).

机译：唐莴苣（Beta vulgaris var。cicla）中过氧化氢酶的纯化和鉴定。
- 作者：Dincer A;Aydemir T
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第2期
- Catalase;
- Chenopodiaceae;
- Chlorides;
- Enzyme Inhibitors;
- Ferric Compounds;
- 过氧化氢酶;
- 藜科;
85.Effects of substrate structural analogues on the enzymatic activities of aspartate aminotransferase isoenzymes.

机译：底物结构类似物对天冬氨酸转氨酶同工酶的酶活性的影响。
- 作者：Martins LL;Mourato MP;de-Varennes A
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- alpha 1-Antitrypsin;
- Donors;
- Isoenzymes;
- -4;
- α1-抗胰蛋白酶;
- 同工酶类;
86.Glycosylasparaginase inhibition studies: competitive inhibitors, transition state mimics, noncompetitive inhibitors.

机译：糖基葡聚糖酶抑制研究：竞争性抑制剂，过渡态模拟物，非竞争性抑制剂。
- 作者：Risley JM;Huang DH;Kaylor JJ;Malik JJ;Xia YQ
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- Aspartylglucosylaminase;
- competition;
- inhibitors;
- VALUING;
- 天冬氨酰葡糖脱氨基酶;
87.Quantitative structure-activity relationship study of novel alpha1a-selective adrenoceptor antagonists.

机译：新型α1a-选择性肾上腺素受体拮抗剂的定量构效关系研究。
- 作者：Singh P;Kumar R
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- structure;
- antagonists;
- novel;
- KAI1 Gene;
- Upper case ecks;
88.Quantitative structure-activity relationships (QSARs) within series of inhibitors for mammalian cytochromes P450 (CYPs).

机译：哺乳动物细胞色素P450（CYPs）抑制剂系列中的定量构效关系（QSAR）。
- 作者：Lewis-D F;Dickins M
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Quantitative Structure-Activity Relationship;
- structure;
- inhibitors;
- lipophilicity;
89.Inhibition of pig liver and Zea mays L. polyamine oxidase: a comparative study.

机译：猪肝和玉米玉米多胺氧化酶的抑制作用：一项比较研究。
- 作者：Federico R;Leone L;Botta M;Binda C;Angelini R;Venturini G;Ascenzi P
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第2期
- Amine Oxidoreductases;
- Corn;
- Enzyme Inhibitors;
- Liver;
- Benzamidines;
- Guanidines;
- 胺氧化还原酶类;
- 玉米;
- 酶抑制剂;
- 肝;
90.Kinetics of inactivation of Ulva pertusa Kjellm alkaline phosphatase by ethylenediaminetetraacetic acid disodium.

机译：乙二胺四乙酸二钠灭活百日草碱性磷酸酶的动力学。
- 作者：Yang D;Wang J;Peng X;An L
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Edetic Acid;
- Ulva;
- kinetic characteristics;
- Enzymes;
- Alkaline Phosphatase;
- 依地酸;
- 酶类;
- 碱性磷酸酶;
91.Isomerase activity of the C-terminal fructose-6-phosphate binding domain of glucosamine-6-phosphate synthase from Escherichia coli.

机译：大肠杆菌的氨基葡萄糖-6-磷酸合酶的C-末端果糖6-磷酸结合域的异构酶活性。
- 作者：Todorova R
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- binding;
- Carbon ion;
- inorganic phosphate;
- Isomerases;
- Glucosamine;
- 异构酶类;
- 葡糖胺;
92.Inhibition of Saccharomyces cerevisiae phosphomannose isomerase by the NO-donor S-nitroso-acetyl-penicillamine.

机译：NO供体S-亚硝基-乙酰基-青霉胺对酿酒酵母磷酸甘露糖异构酶的抑制作用。
- 作者：Salvati L;Mattu M;Tiberi F;Polticelli F;Ascenzi P
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- Saccharomyces cerevisiae;
- Mannose-6-Phosphate Isomerase;
- Donors;
- Penicillamine;
- 酵母菌;
- 酿酒;
- 青霉胺;
93.A new class of potent reversible inhibitors of metallo-proteinases: C-terminal thiol-peptides as zinc-coordinating ligands.

机译：一类新的有效的金属蛋白酶可逆抑制剂：C末端硫醇肽作为锌配位体。
- 作者：Peters K;Jahreis G;Kotters-E M
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Peptides;
- inhibitors;
- Sulfhydryl Compounds;
- Zinc;
- Carbon ion;
- 肽类;
- 巯基化合物;
- 锌;
94.Carbonic anhydrase activity modulators: synthesis of inhibitors and activators incorporating 2-substituted-thiazol-4-yl-methyl scaffolds.

机译：碳酸酐酶活性调节剂：结合了2-取代的噻唑-4-基甲基支架的抑制剂和活化剂的合成。
- 作者：Scozzafava A;Saramet I;Banciu-M D;Supuran-C T
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- AC protocol;
- inhibitors;
- Carbonic Anhydrases;
- Roman Numeral IV;
- sulfamate;
95.Inhibition of succinate-cytochrome C reductase by a ferromacrocyclic complex.

机译：亚铁大环复合物抑制琥珀酸-细胞色素C还原酶。
- 作者：Balbaa M;Khalifa M;el-Sabawaya M;Kandeel K
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第4期
- Psychological inhibition;
- Enzymes;
- Lower case sea;
- succinate;
- Cytochrome c;
- 酶类;
- 细胞色素C;
96.A 3D QSAR study of monoamino oxidase-B inhibitors using the chemical function based pharmacophore generation approach.

机译：使用基于化学功能的药效团产生方法对单氨基氧化酶-B抑制剂进行3D QSAR研究。
- 作者：Gritsch S;Guccione S;Hoffmann R;Cambria A;Raciti G;Langer T
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- inhibitors;
- Chemical compound;
- NOS;
- pharmacophore;
- Type B Monoamine Oxidase;
97.Synthesis and evaluation of dipeptide amides containing N omega-nitroarginine and D-2,4-diaminobutyric acids as inhibitors of neuronal nitric oxide synthase.

机译：包含Nω-硝基精氨酸和D-2,4-二氨基丁酸作为神经元一氧化氮合酶抑制剂的二肽酰胺的合成和评估。
- 作者：Huang H;Martasek P;Roman LJ;Silverman RB
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- Dipeptides;
- Amides;
- Containing;
- inhibitors;
- Neuronal;
- Nitric-Oxide Synthase;
- 二肽类;
- 酰胺类;
- 一氧化氮合酶;
- 氮芥;
98.Evidence for an essential arginine in the flavoprotein nitroalkane oxidase.

机译：黄素蛋白硝基烷氧化酶中必需精氨酸的证据。
- 作者：Gadda G;Banerjee A;Fleming GS;Fitzpatrick PF
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第2期
- Arginine;
- Enzyme Inhibitors;
- Flavoproteins;
- Fusarium;
- Oxygenases;
- Cyclohexanones;
- 精氨酸;
- 酶抑制剂;
- 黄素蛋白类;
- 镰刀菌属;
- 氧合酶类;
99.Structure-activity relationships of new NAPAP-analogs.

机译：新的NAPAP模拟物的构效关系。
- 作者：Steinmetzer T;Schweinitz A;Kunzel S;Wikstrom P;Hauptmann J;Sturzebecher J
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第3期
- New;
- analogs;
- Thrombin;
- 凝血酶;
100.Synthesis and in-vitro evaluation of novel low molecular weight thiocarbamates as inhibitors of human leukocyte elastase.

机译：新型低分子量硫代氨基甲酸酯类化合物作为人白细胞弹性蛋白酶抑制剂的合成及体外评价。
- 作者：Rodis NP;Digenis GA
- 期刊名称：《Journal of enzyme inhibition》 | 2001年第2期

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