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机译:刺参相关蛋白在体内和体外拮抗中枢黑皮质素受体
Department of Pediatrics, Howard Hughes Medical Institute, Stanford University School of Medicine, Stanford, CA 94305, USA.;
Adrenal Glands metabolism; Amino Acid Sequence; Animals; Female; Humans; Hypothalamus metabolism; MSH antagonists inhibitors pharmacology; Male; Melanophores metabolism; Mice; Mice; Inbred C57BL; Mice; Inbred CBA; Mice; Obese; Mice; Transgenic; Molecular Sequence Data; Obesity etiology; Organophosphorus Compounds pharmacology; Proteins chemistry genetics pharmacology physiology; RNA genetics metabolism; Receptor; Melanocortin; Type 3; Receptor; Melanocortin; Type 4; Receptors; Corticotropin antagonists inhibitors metabolism; Receptors; Peptide antagonists inhibitors metabolism; Recombinant Proteins metabolism; Research Support; Non-U.S. Gov't; Research Support; U.S. Gov't; Non-P.H.S.; Research Support; U.S. Gov't; P.H.S.; Signal Transduction; Xenopus;
机译:刺豚鼠相关蛋白和刺豚鼠信号蛋白的环交换嵌合体确定了黑皮质素1受体选择性和拮抗作用所需的接触。
机译:通过体外诱变研究melanocortin-4受体的结构活性:确定刺骨相关蛋白(AGRP),黑皮质素激动剂和合成肽拮抗剂相互作用决定簇。
机译:人类的刺鼠相关蛋白(AGRP)核心十肽(Yc(CRFFNAFC)Y)的延伸研究导致对小鼠黑皮质素3受体的拮抗作用。
机译:与Melanocortin激动剂相比,天然存在的黑色激素拮抗剂agouti相关蛋白(AgrP)具有与MC4受体相似明显的相互作用
机译:在体外和体内研究了乙酰胆碱受体和受体相关的rapsyn支架蛋白的动力学。
机译:刺豚鼠相关蛋白的环已交换嵌合体(agRp的)和刺豚鼠信号蛋白(asIp)确定所需的黑皮素1受体(mC1R)选择性与对抗联系
机译:agouti相关蛋白的环形倒数和agouti信号蛋白鉴定Melanocortin 1受体选择性和拮抗作用所需的触点