机译:USP7小分子抑制剂干扰泛素结合
Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA|Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Struct Biol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Struct Biol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA|Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA|Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA|Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA|Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA;
Univ Dundee, Sch Life Sci, MRC Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland;
Univ Dundee, Sch Life Sci, MRC Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland;
Newcastle Univ, Inst Cell & Mol Biosci, Newcastle Upon Tyne NE2 1HH, Tyne & Wear, England;
Genentech Inc, Dept Prot Chem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Prot Chem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Microchem Prote & Lipid, San Francisco, CA 94080 USA;
Boston Biochem, 840 Mem Dr, Cambridge, MA 02139 USA;
Boston Biochem, 840 Mem Dr, Cambridge, MA 02139 USA;
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA 94143 USA|Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA;
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA 94143 USA|Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA;
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA 94143 USA|Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA;
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA 94143 USA|Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA;
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA 94143 USA|Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA;
Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Microchem Prote & Lipid, San Francisco, CA 94080 USA;
Genentech Inc, Dept Res Pathol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Bioinformat & Computat Biol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Bioinformat & Computat Biol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Bioinformat & Computat Biol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Bioinformat & Computat Biol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Prot Chem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA;
Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA;
Boston Biochem, 840 Mem Dr, Cambridge, MA 02139 USA;
Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Struct Biol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Struct Biol, San Francisco, CA 94080 USA;
Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA|Genentech Inc, Dept Early Discovery Biochem, San Francisco, CA 94080 USA;
机译:使用集成NMR和硅技术发现泛素特异性蛋白酶7(USP7)的小分子抑制剂
机译:鉴定的选择性USP7抑制剂与泛素结合竞争
机译:与Rev1的泛素结合基序结合的小分子抑制Rev1与K164-单突相关PCNA相互作用,抑制DNA损伤耐受性
机译:抗凋亡Bcl-2家族蛋白的广谱小分子抑制剂的设计,合成和活性评估:广谱蛋白结合的特征及其对抗肿瘤活性的影响
机译:HIV-1 gp120:一种新颖的大规模纯化技术和两种小分子抑制剂结合的热力学表征。
机译:结合REV1泛素结合基序的小分子抑制REV1与K164单泛素化PCNA的相互作用并抑制DNA损伤耐受性
机译:USP7小分子抑制剂干扰泛素结合