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Stabilization of G-Quadruplex DNA and Inhibition of Telomerase Activity by Square-Planar Nickel(II) Complexes

机译:G-四链体DNA的稳定和端平面镍(II)配合物抑制端粒酶活性。

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摘要

The enzyme telomerase has an elevated activity in 85-90% of human cancer cells in comparison to normal somatic cells.Telomerase inhibition has thus been identified as an attractive target for cancer chemotherapy with the potential for selective toxicity for cancer cells over normal ones.
机译:与正常的体细胞相比,端粒酶在85-90%的人类癌细胞中具有升高的活性,因此端粒酶抑制作用已被认为是癌症化疗的诱人靶标,与正常细胞相比具有潜在的选择性毒性。

著录项

  • 来源
    《Journal of the American Chemical Society》 |2006年第18期|p.5992-5993|共2页
  • 作者单位

    Department of Chemistry,Imperial College London,South Kensington,London SW7 2AZ,U.K.,CRUK Biomolecular Structure Group,The School of Pharmacy University of London,London WC1N 1AX,U.K.,and Institute of Chemical Research of Catalonia (ICIQ),Avgda.Pai's;

    Department of Chemistry,Imperial College London,South Kensington,London SW7 2AZ,U.K.,CRUK Biomolecular Structure Group,The School of Pharmacy University of London,London WC1N 1AX,U.K.,and Institute of Chemical Research of Catalonia (ICIQ),Avgda.Pai's;

    Department of Chemistry,Imperial College London,South Kensington,London SW7 2AZ,U.K.,CRUK Biomolecular Structure Group,The School of Pharmacy University of London,London WC1N 1AX,U.K.,and Institute of Chemical Research of Catalonia (ICIQ),Avgda.Pai's;

    Department of Chemistry,Imperial College London,South Kensington,London SW7 2AZ,U.K.,CRUK Biomolecular Structure Group,The School of Pharmacy University of London,London WC1N 1AX,U.K.,and Institute of Chemical Research of Catalonia (ICIQ),Avgda.Pai's;

  • 收录信息 美国《科学引文索引》(SCI);美国《工程索引》(EI);美国《生物学医学文摘》(MEDLINE);美国《化学文摘》(CA);
  • 原文格式 PDF
  • 正文语种 eng
  • 中图分类 化学;
  • 关键词

  • 入库时间 2022-08-18 03:22:40

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