机译:端粒G-四链体稳定对化学配体抑制端粒酶介导的端粒延伸的贡献
Laboratory of Biochemistry and Biophysics, College of Life Sciences, Wuhan University, Wuhan 430072, P. R. China;
State Key Laboratory of Biomembrane and Membrane Biotechnology, Institute of Zoology, Chinese Academy of Sciences, Beijing 100101, P. R. China;
Laboratory of Biochemistry and Biophysics, College of Life Sciences, Wuhan University, Wuhan 430072, P. R. China;
State Key Laboratory of Biomembrane and Membrane Biotechnology, Institute of Zoology, Chinese Academy of Sciences, Beijing 100101, P. R. China;
Laboratory of Biochemistry and Biophysics, College of Life Sciences, Wuhan University, Wuhan 430072, P. R. China,State Key Laboratory of Biomembrane and Membrane Biotechnology, Institute of Zoology, Chinese Academy of Sciences, Beijing 100101, P. R. China;
机译:分子拥挤条件下端粒G-四链体的稳定性降低或减弱,端粒酶被小化学配体抑制。
机译:端粒相关蛋白的表达是相互依赖的,以稳定天然端粒结构和G-Quadreplex配体的端粒功能障碍导致Terra Upregulation
机译:N-环湾取代的G G-四链体配体系列中的芳香核心扩展:端粒损伤增加,抗肿瘤活性和对健康细胞的肿瘤的强选择性。
机译:具有可调谐侧链的新型四龙布雷宏γ作为G-Quadreplex稳定配体
机译:靶向端粒G-四链体的全长端粒悬突中形成的二级结构和配体的合理设计研究。
机译:端粒和端粒酶相互作用蛋白可在哺乳动物细胞中展开端粒G-四链体并促进端粒延伸
机译:内部封面:寻找有效的G-quadruplex配体:用于使用药物状分子选择性稳定性质和端粒损伤的证据(ChemMedchem 4/2015)