机译:Eudistidine A的结构阐明和合成:一种异常的多环海洋生物碱,其阻断p300和HIF-1α的蛋白质结合域的相互作用。
Molecular Targets Laboratory, Center for Cancer Research, National Cancer Institute, Frederick, Maryland 21702-1201, United States;
Chemical Biology Laboratory, Center for Cancer Research, National Cancer Institute, Frederick, Maryland 21702-1201, United States,National Center for Advancing Translational Sciences, National Institutes of Health, Bethesda, Maryland 20892, United States;
Molecular Targets Laboratory, Center for Cancer Research, National Cancer Institute, Frederick, Maryland 21702-1201, United States;
Molecular Targets Laboratory, Center for Cancer Research, National Cancer Institute, Frederick, Maryland 21702-1201, United States,Basic Science Program, Leidos Biomedical Research, Inc., Frederick National Laboratory for Cancer Research, Frederick, Maryland 21702-1201, United States;
Molecular Targets Laboratory, Center for Cancer Research, National Cancer Institute, Frederick, Maryland 21702-1201, United States,Diagnostic Biomarkers and Technology Branch, Cancer Diagnosis Program, DCTD, National Cancer Institute, Bethesda, Maryland 20850, United States;
Genitourinary Malignancies Branch, Center for Cancer Research, National Cancer Institute, Bethesda, Maryland 20892, United States;
Genitourinary Malignancies Branch, Center for Cancer Research, National Cancer Institute, Bethesda, Maryland 20892, United States;
Genitourinary Malignancies Branch, Center for Cancer Research, National Cancer Institute, Bethesda, Maryland 20892, United States;
Molecular Targets Laboratory, Center for Cancer Research, National Cancer Institute, Frederick, Maryland 21702-1201, United States;
Chemical Biology Laboratory, Center for Cancer Research, National Cancer Institute, Frederick, Maryland 21702-1201, United States;
Molecular Targets Laboratory, Center for Cancer Research, National Cancer Institute, Frederick, Maryland 21702-1201, United States;
机译:海洋吡咯烷氨基醌生物碱的筛选和生物效应:HIF-1 alpha / p300相互作用的潜在抑制剂。
机译:包含炔基和链烷烃呋喃的噻唑烷酮破坏HIF-1 alpha和p300蛋白相互作用的设计,合成和生物活性评估
机译:Eudistidine C的表征和合成,具有生物分子支架的生物活性海洋生物碱。
机译:Pichia牧场表达系统中融合蛋白的MBP(麦芽糖结合蛋白)C-末端的结构阐明
机译:质谱法以阐明蛋白质 - 蛋白质相互作用,牙买蛋白域的生化和结构表征,以及带3作为红细胞代谢和储存质量的主调节器的作用
机译:Eudistidine A的结构阐明和合成:一种异常的多环海洋生物碱其阻断p300和HIF-1α的蛋白质结合域的相互作用。
机译:小泛素样修饰蛋白1(sUmO1)与CREB结合蛋白ZZ结构域(CBp / p300)之间复合物的结构分析揭示了sUmO上新的相互作用表面