National-Local Joint Engineering Laboratory of Druggability and New Drugs Evaluation;
Guangdong Province Engineering Laboratory for Druggability and New Drugs Evaluation;
School of Pharmaceutical Sciences;
Sun Yat-sen University;
Guangzhou 510006;
China;
G proteins; Gaq/11 inhibitors; SARs; BRET; Uveal melanoma; Antitumor; Safety; Pharmacokinetics;