首页> 外国专利> Hydrochloride Salt of (1S, 2S, 4R) - 4 - (4 - (1S) - 2,3 dihydro - 1 - 1 - ilamino inden - - 7h pyrrolo 2,3-d pyrimidine 7 - il} - 2 - hidroxiciclopentil) metilsulfamato

Hydrochloride Salt of (1S, 2S, 4R) - 4 - (4 - (1S) - 2,3 dihydro - 1 - 1 - ilamino inden - - 7h pyrrolo 2,3-d pyrimidine 7 - il} - 2 - hidroxiciclopentil) metilsulfamato

机译:(1S,2S,4R)-4-(4-[(1S)-2,3 dihydro-1-1-ilamino inden-]-7h pyrrolo [2,3-d]嘧啶7-il}-的盐酸盐2-广西氯喷地(metilsulfamato)

摘要

It refers to a Crystal hydrochloride ((1S, 2S, 4R) - 4 - (4 - [(1S) - 2,3 dihydro - 1 - 1 - ilamino inden -] - 7h pyrrolo [2,3-d] pyrimidine 7 - il} - 2 - hidroxiciclopentil) characterized by metilsulfamato formula I a pattern that has 2 Peaks XRPD Angle (Theta): 7.3u00ba, 9.6u00ba, 13.6u00ba, 14.5u00ba, 14.8u00ba, 16.5u00ba, 17.0u00ba, 17.3u00ba, 18.0u00ba, 19.1u00ba, 20.1u00ba, 21.1u00ba, 21.7u00ba, 23.7u00ba + - 0.2 degrees.It also relates to a production method and a Pharmaceutical formulation. The Glass is an inhibitor of E1 Activating Enzyme, being useful in the treatment of cancer
机译:它是指晶体盐酸盐((1S,2S,4R)-4-(4-[(1S)-2,3二氢-1-1-氨基氨基茚满-]-7h吡咯并[2,3-d]嘧啶7 -il}-2-盐酸西地罗非尼(i),其特征在于metilsulfamato分子式I具有2个峰的XRPD角(θ)的模式:7.3 u00ba,9.6 u00ba,13.6 u00ba,14.5 u00ba,14.8 u00ba,16.5 u00ba,17.0所述玻璃是一种制备方法和药物制剂,其为1°C,17.3°C,18.0°C,10.1°C,20.1°C,21.1°C,21.7°C,23.7°C,23.7°C + -0.2度。 E1活化酶抑制剂,可用于治疗癌症

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