首页> 外国专利> PHARMACEUTICAL COMPOSITION, METHOD FOR PREPARING THE SAME, METHODS FOR INHIBITING THE RATE AGENT PRECIPITATION RATE, AND FOR REDUCING INTERPATIENT VARIABILITY WITH REGARD TO BIODISPONIBILITY AND / OR CONCENTRATION, AND / OR CONCENTRATION WATER SOLUBLE Aether CELLULOSE OR AN ESTER OF A WATER SOLUBLE ETHER CELLULOSE

PHARMACEUTICAL COMPOSITION, METHOD FOR PREPARING THE SAME, METHODS FOR INHIBITING THE RATE AGENT PRECIPITATION RATE, AND FOR REDUCING INTERPATIENT VARIABILITY WITH REGARD TO BIODISPONIBILITY AND / OR CONCENTRATION, AND / OR CONCENTRATION WATER SOLUBLE Aether CELLULOSE OR AN ESTER OF A WATER SOLUBLE ETHER CELLULOSE

机译:药物组合物,制备该药物的方法,抑制速率剂沉淀率的方法以及用于降低生物相容性和/或浓度和/或浓度的水溶性硅藻土,纤维素,纤维素,纤维素,纤维素或酯类化合物之间的差异的方法

摘要

"pharmaceutical composition, method for preparing same, methods for inhibiting the precipitation agent of the solution agent in the GI tract, and for reducing inter-patient variability with respect to bioavailability and / or plasma concentrations of the agent, and use of a water soluble ether cellulose or an ester of a water soluble ether cellulose ". a pharmaceutical composition comprising 4- (3'-chloro-4'-fluoroanilino) -7-methoxy-6- (3-morpholine-propoxy) quinazoline or a pharmaceutically acceptable salt thereof (the agent) and a soluble ether cellulose in water or an ester of a water-soluble ether cellulose. Water soluble ether cellulose or ester of a water soluble ether cellulose present in the composition inhibits the precipitation rate of the solution agent.
机译:“药物组合物,其制备方法,抑制胃肠道中溶液剂沉淀剂的方法,以及减少患者在药物的生物利用度和/或血浆浓度方面的差异的方法,以及水溶性醚纤维素或水溶性醚纤维素的酯”。药物组合物,其包含4-(3'-氯-4'-氟苯胺基)-7-甲氧基-6-(3-吗啉-丙氧基)喹唑啉或其药学上可接受的盐(该试剂)和在水中的可溶性醚纤维素或水溶性醚纤维素的酯。组合物中存在的水溶性醚纤维素或水溶性醚纤维素的酯抑制溶液剂的沉淀速率。

著录项

  • 公开/公告号BRPI0307786B1

    专利类型

  • 公开/公告日2018-03-13

    原文格式PDF

  • 申请/专利权人 ASTRAZENECA AB;

    申请/专利号BR2003PI07786

  • 申请日2003-02-24

  • 分类号A61K9/16;A61K47/38;A61K;A61K9/10;A61K9/20;A61K9/28;A61K31/517;A61K31/5377;A61K47/20;A61K47/32;A61K47/36;A61P35;A61P43;C07D239/94;

  • 国家 BR

  • 入库时间 2022-08-21 12:53:26

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