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机译:Dichloro Butenediamides as Irreversible Site-Selective Protein Conjugation Reagent
Univ Cambridge, Yusuf Hamied Dept Chem, Lensfield Rd, Cambridge CB2 1EW, England;
Scripps Res Inst, Dept Chem, 130 Scripps Way, Jupiter, FL 33458 USA;
Univ Lisbon, Inst Med Mol Joao Lobo Antunes, Fac Med, Ave Prof Egas Moniz, P-1649028 Lisbon, PortugalAstraZeneca, Antibody Discovery & Prot Engn ADPE, R&D BioPharmaceut Unit, Milstein Bldg,Granta Pk, Cambridge CB21 6GH, EnglandUniv La Rioja, Ctr Invest Sintesis Quim, Dept Quim, Logrono 26006, Spain;
bioconjugation; cysteine; irreversibility; maleimides; Michael addition;