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机译:通过靶向非保守的残留物和结构性水位移选择性N-末端下注溴染色剂**
Univ Minnesota Twin Cities Dept Chem 207 Pleasant St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Med Chem 2231 6th St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Chem 207 Pleasant St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Chem 207 Pleasant St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Chem 207 Pleasant St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Chem 207 Pleasant St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Chem 207 Pleasant St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Biochem Mol Biol &
Biophys 321 Church St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Biochem Mol Biol &
Biophys 321 Church St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Med Chem 2231 6th St SE Minneapolis MN 55455 USA;
Univ Minnesota Twin Cities Dept Chem 207 Pleasant St SE Minneapolis MN 55455 USA;
BET bromodomains; BRD4 D1 selectivity; epigenetics; inhibitors; structure-activity relationships;
机译:基于结构的溴琼肿瘤域(BET)抑制剂选择性,用于保留抗炎和抗增殖表型的N-末端溴染色剂
机译:PFI-1,一种高度选择性的蛋白质相互作用抑制剂,靶向BET溴结构域
机译:ZA通道水介导的相互作用在溴琼域选择性BET抑制剂设计中的作用
机译:(8)污泥生产在钝化涂层和抑制酸性矿井水中产生的污泥生产
机译:靶向Hsp90的两端:嵌合的N末端抑制剂和新霉素衍生的C末端抑制剂。
机译:ZA通道水介导的相互作用在溴结构域选择性BET抑制剂设计中的作用
机译:通过靶向非保守的残留物和结构水位,有效和选择性N末端BRD4溴染色剂
机译:BET Bromodomain抑制剂在乳腺癌中的作用机制。